Arecaidine | Arecaidine But-2-Ynyl Ester Tosylate | GABA Uptake Inhibitor

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槟榔次碱 /Arecaidine 99%+

货号：A347338 同义名： Arecaidine But-2-Ynyl Ester Tosylate

Arecaidine but-2-ynyl ester tosylate is a potent muscarinic agonist that shows 4.6-fold that is selectivity for mAChR M2 in the atrium versus those in the ileum.

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Type	HazMat fee for 500 gram (Estimated)
Excepted Quantity	USD 0.00
Limited Quantity	USD 15-60
Inaccessible (Haz class 6.1), Domestic	USD 80+
Inaccessible (Haz class 6.1), International	USD 150+
Accessible (Haz class 3, 4, 5 or 8), Domestic	USD 100+
Accessible (Haz class 3, 4, 5 or 8), International	USD 200+

Arecaidine 化学结构
CAS号：499-04-7

Arecaidine 3D分子结构
CAS号：499-04-7

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Arecaidine 纯度/质量文件产品仅供科研

货号：A347338 标准纯度： 99%+ 产品说明书

批次查询：批次纯度: COA SDS NMR HPLC CNMR LC-MS

全球学术期刊中引用的产品: • Nat. Commun., 2024, 15, 7687. Ambeed. [ A119633 ]; • ACS Nano, 2024. Ambeed. [ A1194179 ]; • J. Mol. Cell. Cardiol., 2024, 196, 94-104. Ambeed. [ A133052 ]; • iScience, 2024, 110928. Ambeed. [ A1375212 ]; • Mol. Pharmaceutics, 2024. Ambeed. [ A305202 , A409401 ]; 更多 >

AChR 亚型比较

产品名称	AChE ↓ ↑	AChR ↓ ↑	mAChR ↓ ↑	nAChR ↓ ↑	其他靶点	纯度
Donepezil	+++ bAChE, IC50: 8.12 nM hAChE, IC50: 11.6 nM					98%
Loganin	++ AChE, IC50: 3.95 μM					99%+
topride HCl	++ AChE, IC50: 2.04 μM					98%
Dehydroevodiamine HCl	✔					99%+
Jatrorrhizine	++ AChE, IC50: 872 nM					99%+
Palmatine	++ AChE, IC50: 0.51 μM					98%
(-)-Huperzine A	++++ AChE (G4 form), Ki: 7 nM					98%
Galanthamine HBr	++ AChE, IC50: 0.35 μM					98%
Trospium chloride		✔				99%
Tiotropium Bromide Monohydrate		✔				98+%
Gallamine Triethiodide		+ AChR, IC50: 68.0 μM				98%
Hexamethonium Bromide		✔				99%
Pancuronium dibromide		✔				98%
Neostigmine bromide		✔				98%
Orphenadrine citrate		✔				98%
Oxybutynin		✔				98%
Irsogladine		✔			PDE	98%
Pyridostigmine bromide		✔				99+%
Rivastigmine		+ AChR, IC50: 5.5 μM				98%
Paroxetine hydrochloride		✔				97%
Rocuronium Bromide		✔				98%
Tropicamide			+++ M4 mAChR, IC50: 8 nM			98%
Diphenmanil methylsulfate			✔			98%
Umeclidinium bromide			✔			95%
Otilonium bromide			✔			98%
Flavoxate HCl			+ mAChR, IC50: 12.2 μM			98%
Ipratropium bromide			✔			98%
Diphenidol HCl			✔			98%
Darifenacin hydrobromide			++++ M3 mAChR, pKi: 8.9			98%
Aclidinium Bromide			++++ M4 mAChR, Ki: 0.21 nM M2 mAChR, Ki: 0.1 nM			98%
Oxybutynin chloride			✔			99%
Pentoxyverine citrate			✔			98%
Solifenacin			✔			98%
Catharanthine				✔		98%
Benzethonium chloride				+++ α7 nAChRs, IC50: 122 nM α4β2 nAChRs, IC50: 49 nM		99+%
Vinblastine sulfate				+ nAChR, IC50: 8.9 μM		99%
PNU-120596				++ α7 nAChR, EC50: 216 nM		99+%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。

Arecaidine 生物活性

描述	Arecaidine but-2-ynyl ester tosylate is a potent muscarinic agonist that shows 4.6-fold that is selectivity for mAChR M2 in the atrium versus those in the ileum.

Arecaidine 参考文献

[1]Moser U, Lambrecht G, et al. Structure-activity relationships of new analogues of arecaidine propargyl ester at muscarinic M1 and M2 receptor subtypes. Br J Pharmacol. 1989 Feb;96(2):319-24.

[2]Barlow RB, Weston-Smith P. The relative potencies of some agonists at M2 muscarinic receptors in guinea-pig ileum, atria and bronchi. Br J Pharmacol. 1985 Jun;85(2):437-40.

Arecaidine 实验方案

计算器

存储液制备

1mg

5mg

10mg

1 mM

5 mM

10 mM

7.08mL

1.42mL

0.71mL

35.42mL

7.08mL

3.54mL

70.84mL

14.17mL

7.08mL

Arecaidine 技术信息

CAS号	499-04-7
分子式	C₇H₁₁NO₂
分子量	141.168

别名	Arecaidine But-2-Ynyl Ester Tosylate
运输	蓝冰

存储条件

粉末 Sealed in dry,2-8°C

液体 -20°C:3-6个月-80°C:12个月

溶解度

H₂O: 250 mg/mL(1770.94 mM)，配合低频超声助溶

动物实验配方

槟榔次碱 /Arecaidine 99%+

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槟榔次碱 /Arecaidine 99%+

Arecaidine 纯度/质量文件 产品仅供科研

全球学术期刊中引用的产品

Arecaidine 质控信息

Arecaidine 生物活性

Arecaidine 参考文献

Arecaidine 实验方案

Arecaidine 技术信息

最近浏览的产品

大规格询价

摩尔计算器

靶点

总药量计算器

工作液计算器

细胞研究

临床研究

确认信息

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热门区域

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B

C

F

G

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J

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Arecaidine 纯度/质量文件产品仅供科研