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Centanafadine HCl
Centanafadine HCl
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货号：A1177284
同义名：
EB-1020 hydrochloride;Centanafadine hydrochloride
Centanafadine HCl是一种双重去甲肾上腺素 (NE) 和多巴胺 (DA) 转运抑制剂，同时对 5-羟色胺转运体也有抑制作用。其对 NE、DA 和 5-HT 转运体的 IC50 值分别为 6 nM、38 nM 和 83 nM，适用于注意缺陷多动障碍 (ADHD) 及其他神经系统疾病的研究。
Centanafadine HCl 化学结构
CAS号：923981-14-0
Centanafadine HCl 3D分子结构
CAS号：923981-14-0
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Centanafadine HCl 纯度/质量文件 产品仅供科研
货号：A1177284
标准纯度：
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Centanafadine HCl 质控信息
| Penfluridol |
+
Dopamine receptor, Ki: 1.6 μM
|
|
|
|
|
|
|
|
98% |
| Ansofaxine HCl |
++
Dopamine receptor, IC50: 491 nM
|
|
|
|
|
|
|
|
99% |
| Tetrahydroberberine,THB |
|
+
|
|
|
|
|
|
|
98+% |
| Prochlorperazine Maleate |
|
✔
|
|
|
|
|
|
|
98% (HPLC) |
| Olanzapine |
|
✔
|
|
|
|
|
|
|
99+% |
| Trifluoperazine |
|
++++
Dopamine D2 receptor, IC50: 1.1 nM
|
|
|
|
|
|
|
98% |
| Ropinirole hydrochloride |
|
++
|
|
|
|
|
|
|
99% |
| Lurasidone |
|
++++
|
|
|
|
|
|
|
98% |
| Levosulpiride |
|
✔
|
|
|
|
|
|
|
99+% |
| Pridopidine |
|
✔
|
|
|
|
|
|
|
95% |
| Metoclopramide |
|
✔
|
|
|
|
|
✔
|
|
99+% |
| Molindone HCl |
|
✔
|
|
|
|
|
|
|
99% |
| Sulpiride |
|
✔
|
|
|
|
|
|
|
99+% |
| Perospirone |
|
++++
|
|
|
|
|
|
|
99% |
| Perospirone HCl |
|
++++
|
|
|
|
|
|
|
99% |
| Phenothiazine |
|
✔
|
|
|
|
|
|
|
98% |
| Pimozide |
+
Dopamine D1 receptor, Ki: 6600 nM
|
+++
Dopamine D2 receptor, Ki: 3.0 nM
|
++++
Dopamine D3 receptor, Ki: 0.83 nM
|
|
|
|
|
|
98% |
| Rotundine |
++
D1 receptor, IC50: 166 nM
|
+
D2 receptor, IC50: 1.47 μM
|
+
D3 receptor, IC50: 3.25 μM
|
|
|
|
|
|
98% |
| Domperidone |
|
✔
|
|
|
|
|
|
|
99+% |
| ONC206 |
|
✔
|
|
|
|
|
|
|
99% |
| Pimethixene maleate |
++
Dopamine D1 Receptor, pKi: 6.37
|
+++
Dopamine D2 Receptor, pKi: 8.19
|
|
++
Dopamine D4.4 Receptor, pKi: 7.54
|
|
|
|
|
97% |
| Loxapine succinate |
++
D2 receptor (Human), Ki: 62 nM
D1 receptor (human), Ki: 26 nM
|
++
D2 receptor (human), Ki: 24 nM
D2 receptor (bovine), Ki: 26 nM
|
|
+++
D4 receptor (human), Ki: 7.5 nM
|
|
|
|
|
99% |
| Chlorprothixene |
+++
|
+++
|
+++
|
|
+++
|
|
|
|
99% |
| SCH-23390 HCl |
++++
D1 dopamine receptor, Ki: 0.2 nM
|
|
|
|
++++
D5 dopamine receptor, Ki: 0.3 nM
|
|
|
|
98% |
| MPP+ iodide |
|
|
|
|
|
✔
|
|
|
97% |
| σ1 Receptor antagonist-1 |
|
|
|
|
|
+
|
|
|
97% |
| Benztropine mesylate |
|
|
|
|
|
++
|
|
|
98% |
| Azaperone |
|
|
|
|
|
|
✔
|
|
98% |
| Ziprasidone HCl |
|
|
|
|
|
|
✔
|
|
98+% |
| Paliperidone |
|
|
|
|
|
|
✔
|
|
98% |
| Alizapride HCl |
|
|
|
|
|
|
✔
|
|
99+% |
| Amisulpride |
|
|
|
|
|
|
✔
|
|
98% |
| Quetiapine hemifumarate |
|
|
|
|
|
|
✔
|
Adrenergic Receptor
|
98% |
| Clozapine N-oxide |
|
|
|
|
|
|
✔
|
|
99% |
|
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
|
| Ivabradine HCl |
✔
|
|
|
|
98% |
| Maprotiline hydrochloride |
✔
|
|
|
|
98% |
| Cisatracurium besylate |
✔
|
|
|
|
96% |
| Yohimbine HCI |
|
✔
|
|
|
99+% |
| BMY 7378 |
|
++
α1D-adrenoceptor, pKi: 5.1
α2C-adrenoceptor, pKi: 6.54
|
+
β1-adrenoceptor, pIC50: 5.1
|
|
97% |
| Asenapine maleate |
|
++++
α2A-adrenergic receptor, pKi: 8.9
α2B-adrenergic receptor, pKi: 8.9
|
|
|
97% |
| Piribedil |
|
++
adrenoceptor α2A, pKi: 7.1
adrenoceptor α2C, pKi: 7.2
|
|
|
98% |
| Prazosin HCl |
|
✔
|
|
|
95% |
| Silodosin |
|
✔
|
|
|
98% |
| Phenoxybenzamine HCl |
|
✔
|
|
|
98% |
| Naftopidil |
|
+++
α1A-adrenergic receptor, Ki: 3.7 nM
α1D-adrenergic receptor, Ki: 20 nM
|
|
|
98% |
| Naftopidil 2HCl |
|
+
α1-adrenergic receptor, IC50: 0.2 μM
|
|
|
99% |
| Alfuzosin HCl |
|
✔
|
|
|
98% |
| Terazosin HCl |
|
✔
|
|
|
99% |
| Atipamezole |
|
✔
|
|
|
95% |
| Phentolamine methanesulfonate salt |
|
✔
|
|
|
99% |
| Doxazosin mesylate |
|
✔
|
|
|
99% |
| Tolazoline HCl |
|
✔
|
|
|
98% |
| Zenidolol hydrochloride |
|
|
++++
β2-adrenergic receptor, Ki: 0.7nM
β1-adrenergic receptor, Ki: 611nM
|
|
98% |
|
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
|
Centanafadine HCl 实验方案
| 计算器 |
|
| 存储液制备 |
 |
1mg |
5mg |
10mg |
|
1 mM
5 mM
10 mM
|
4.07mL
0.81mL
0.41mL
|
20.35mL
4.07mL
2.03mL
|
40.69mL
8.14mL
4.07mL
|
Centanafadine HCl 技术信息
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