匹美噻吨马来酸盐 /Pimethixene maleate
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货号：A293853
同义名：
Pimetixene maleate
Pim ethixene maleate
Pimethixene maleate 化学结构
Pimethixene maleate 3D分子结构
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Pimethixene maleate 纯度/质量文件 产品仅供科研
货号：A293853
标准纯度：
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产品说明书
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Pimethixene maleate 质控信息
Hydroxyzine 2HCl
99+%
Cyclizine
✔
97%
Loratadine
+
98%
Desloratadine
++
Histamine H1 receptor, IC50: 51 nM
98%
Doxylamine succinate
✔
99%
Ebastine
✔
98%
Tripelennamine HCl
+
98%
Meclizine dihydrochloride
✔
98%
Chlorpheniramine maleate
+++
Histamine H1 receptor, IC50: 12 nM
99%
Diphenhydramine HCl
✔
99%
Alcaftadine
++++
++
99%+
Fexofenadine HCl
++
Histamine H1 receptor, IC50: 246 nM
99%+
Bilastine
+++
H1 receptor, Ki: 44.15 nM
98%
Pemirolast potassium
✔
98%
Bepotastine besilate
+
Histamine H1 receptor, pIC50: 5.7
98%
Mizolastine
+++
Histamine H1 receptor, IC50: 47 nM
98%
Brompheniramine maleate
✔
98%
Carbinoxamine maleate salt
✔
99+%
Clemastine fumarate
++++
Histamine H1 receptor, IC50: 3 nM
98%
Ketotifen fumarate salt
✔
95%
Rupatadine Fumarate
++
Histamine H1 receptor, Ki: 102 nM
PAFR
98%
Famotidine
✔
97%
Roxatidine Acetate HCl
+
Histamine H2 receptor, IC50: 3.2 μM
98%
Lafutidine
✔
99%
Cimetidine
✔
98%
Nizatidine
++++
Histamine H2 receptor, IC50: 0.9 nM
AChE
98%
Ranitidine
✔
99%
Betahistine
+
Histamine H3 receptor, IC50: 1.9 μM
98%
Ciproxifan maleate
+++
Histamine H3 receptor, IC50: 9.2 nM
99%+
S 38093
++
human H3 receptor, Ki: 1.2 μM
rat H3 receptor, Ki: 1.44 μM
98%
JNJ-7777120
++++
Histamine H4 receptor, Ki: 4.5 nM
98%
Azelastine HCl
✔
98%
Epinastine HCl
✔
98%
Levodropropizine
✔
97%
Cyproheptadine hydrochloride
✔
98%
Hesperetin
✔
97%
Olopatadine HCl
✔
98%
Mianserin hydrochloride
✔
99+%
Buclizine 2HCl
✔
97%
Latrepirdine 2HCl
✔
GluR
98%
Cetirizine 2HCl
✔
98%
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1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
Pimethixene maleate 生物活性
靶点
D4 receptor
Dopamine D4.4 Receptor, pKi:7.54
D1 receptor
Dopamine D1 Receptor, pKi:6.37
D2 receptor
Dopamine D2 Receptor, pKi:8.19
描述
Similarly, Pimethixene maleate acts as both an antihistamine and an antiserotonergic compound, also used for migraine prevention. It antagonizes the same receptors as Pimethixene with identical potency and binding affinities[1]
Pimethixene maleate 参考文献
Pimethixene maleate 实验方案
计算器
摩尔计算器
总药量计算器
工作液计算器
存储液制备
1mg
5mg
10mg
1 mM
5 mM
10 mM
2.44mL
0.49mL
0.24mL
12.21mL
2.44mL
1.22mL
24.42mL
4.88mL
2.44mL
Pimethixene maleate 技术信息
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