Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.

JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.

Landiolol hydrochloride (ONO1101 hydrochloride) is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity = 255:1, a half-life of 4 min)， acts as an adrenoceptor antagonist[1].

Terazosin HCl is an α-adrenergic (AL-fa ad-ren-ER-jik) blocker used in the therapy of hypertension and benign prostatic hypertrophy with climination half-life‎ of ‎12 hours.

Tolazoline HCl is a competitive non-selective α-adrenergic receptor antagonist, used as a a vasodilator directly acting on blood vessels and also increasing cardiac output.

Nicergoline is a non-selective alpha-adrenergic receptor antagonist which can decrease vascular resistance and increase arterial blood flow in the brain, improving the utilization of oxygen and glucose by brain cells.

Medetomidine is an agonist of α2-adrenoceptor with Ki value of 1.08 nM, used as both a surgical anesthetic and analgesic.

Scopine HCl salt is a naturally occuring α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock and also s a potential brain-targeting moiety for enhancing the brain uptake efficiency of chlorambucil.

Vibegron是一种有效的、选择性 β3-肾上腺素能受体激动剂 (EC₅₀=1.1 nM)，主要用于治疗膀胱过度活动症及严重急症尿失禁，具有显著的治疗效果。

Carazolol-d7是 Carazolol 的氘代同位素标记物，常用于药代动力学研究，帮助探究 Carazolol 的代谢途径。

Practolol是一种选择性 β1 肾上腺素能受体拮抗剂，可用于心律失常研究。

Romifidine是一种 α2 肾上腺素受体激动剂，表现出显著的镇静作用，广泛用于麻醉及疼痛管理，特别是在动物模型中的应用较为常见。

Meranzin, a natural product isolated and purified from the peel of Citrus maxima, can induce similar effect to Fructus Aurantii on intestinal motility and it was, at least in part, mediated by stimulation of H1 histamine receptors.

BMY 14802是一种 sigma-1 受体 (σ1R) 的拮抗剂，同时也是 5-HT 1A 受体和 α-1 肾上腺素能受体的激动剂。该化合物在帕金森病 (PD) 的大鼠模型中可抑制异常不自主运动 (AIM)，并下调其表达，适用于帕金森病的研究。

Harmane是一种β-咔啉生物碱，具有显著的神经毒性及MAO A/B抑制活性，适用于研究神经毒性、MAO抑制和相关生物学过程。

Clozapine-d8是Clozapine的氘代同位素化合物。Clozapine 是一种抗精神病药物，具有高效结合多种神经受体的能力，广泛用于精神分裂症的研究。

Isorhoifolin is a natural product isolated and purified from the leaves of Citrus paradisi. with weak anti-H2O2 features, antiradical, anti-hyperpermeability, anti-inflammatory and anticancer actions in vitro and in vivo.

Phentolamine是一种选择性的 α1 和 α2 肾上腺素受体 (AR) 拮抗剂，通过阻断这些受体可引起血管扩张。它已被用于勃起功能障碍的研究和治疗，能够逆转血管收缩，改善阴茎的血液流动，表现出良好的抗勃起功能障碍效果。

Propafenone (SA-79) 是一种钠通道阻滞剂，具有抗心律失常作用。它还对β受体具有高亲和力（IC50=32 nM）。Propafenone通过诱导线粒体功能障碍和凋亡抑制食管癌增殖。

(Rac)-Rotigotine (N-0437) 是 Rotigotine 的外消旋体，是多巴胺受体激动剂，部分激动 5-HT1A 受体，并拮抗 α2B-肾上腺素受体。