BRD4 (1), IC50: 77 nM

BRD4 (2), IC50: 33 nM

BRD3, IC50: 0.25 μM

BRD4, IC50: 0.5 μM

BET proteins, IC50: 35 nM

BRD4, pIC50: 5.3

BRD9, pIC50: 7.3

BRD7, IC50: 117 nM

BRD9, IC50: 19 nM

BRD4-BD1, IC50: 39 nM

BRD4 BD2, Kd: 28 nM

BRD4 BD1, Kd: 90 nM

BRD4, Kd: 37 nM

BRD2, IC50: 0.29 μM

BRD9, IC50: 0.122 μM

CECR2, IC50: 17 nM

BRD4 (1), Kd: 170 nM

BRD9, Kd: 5.9 nM

BRD7, Kd: 73 nM

CECR2, Kd: 77 nM

FL-BRD4, IC50: 5 nM

BRD4 BD2, Kd: 1.7 nM

BRD3 BD1, Kd: 2.1 nM

BRD4(1), IC50: 0.43 μM

BRD4, IC50: 14 nM

BRD4, IC50: 20 nM

Brd2(BD2), Kd: 62 nM

Brd3(BD2), Kd: 13 nM

BRD4_BD1, DC50: 500 nM

BRD4, IC50: 241 nM

BRD3-BD1, IC50: 9 nM

BRD4-BD1, IC50: 119 nM

BRD4 BD1, IC50: 27 nM

BRD4 BD2, IC50: 32 nM

BRD4-BD2, IC50: 41 nM

BRD4-BD1, IC50: 5 nM

BRD4 (1), Kd: 82 nM

BRD2-BD1, IC50: 75nM

BRD4-BD1, IC50: 143 nM

BRD42, IC50: 3070 nM

BRD41, IC50: 3070 nM

BRD3_BD2, IC50: 98 nM

BRD4_BD2, IC50: 214 nM

BRD9, DC50: 3 nM

BAZ2A, Kd: 257 nM

BAZ2B, Kd: 136 nM

L3MBTL4, IC50: 6 μM

L3MBTL3, IC50: 35 μM

SMARCA2A, Kd: 72 nM

SMARCA4, Kd: 55 nM

L3MBTL3- D274A, IC50: 3.5 μM

L3MBTL3, IC50: 120 nM

EED, Kd: 82 nM

PRC2, Kd: 114 nM

L3MBTL1, Kd: 3.9 μM

CREB, IC50: 81 nM

EED, IC50: 247 nM

BAZ1A, Kd: 0.52 μM

BRPF2, IC50: 7.9 μM

BRPF1, IC50: 80 nM

BRPF2, Kd: 500 nM

BRPF1B, Kd: 100 nM

BRPF2, pIC50: 5.2

BRPF3, pIC50: 7.1

BRPF1, pIC50: 8.1

BRPF1, IC50: 48 nM

BRPF3, IC50: 260 nM

CBP/beta-catenin, IC50: 0.0484 μM

CBP, Kd: 151 nM

p300, Kd: 167 nM

p300, IC50: 5 μM

p300/CBP, Ki: 400 nM

PCAF, IC50: 5 μM

p300/CBP, IC50: 8.5 μM

EP300, IC50: 38 nM

CREBBP, IC50: 21 nM

p300, IC50: ~25 μM

CREBBP, IC50: 125nM

p300/CBP, IC50: 363nM

EP300, IC50: 0.051 μM

CBP, IC50: 0.03 μM

p300 HAT, IC50: 0.06 μM

BRD4(1), IC50: 5100 nM

CBP, IC50: 0.94 nM

BET, IC50: <30 nM

p300/CBP, IC50: <30 nM

STAT3, IC50: 4.6 μM

STAT3, IC50: 5.1 μM

STAT3, IC50: 86 μM

STAT3, Kd: 4.7 nM

STAT3, Kd: 300 nM

STAT5, Kd: 464 nM