GRI977143是一种特异性 LPA2 受体激动剂，EC50 为 3.3 μM。

Azoramide is a modulator of the unfolded protein response (UPR) with antidiabetic activity.

Boc-Asp(OMe)-fluoromethyl ketone是一种广泛的 caspase 抑制剂，可抑制 Fas 介导的吞噬作用和氧化破裂抑制，但不影响 IL-8 的趋化活性。该化合物在研究细胞凋亡及相关免疫反应中具有潜在应用价值。

Raptinal 直接激活 caspase-3，启动 caspase 依赖的内在凋亡途径。Raptinal 可以通过直接激活效应 caspase-3 快速诱导癌细胞死亡，绕过 initiator caspase-8 和 caspase-9 的激活。

Ac-DEVD-CHO是一种特异性的Caspase-3抑制剂，Ki值为230 pM。

Alisol B is a natural product isolated and purified from the tubers of Alisma plantago-aquatica Linn. for bone disorders by targeting the differentiation of osteoclasts as well as their functions.

Ivachtin (Caspase-3 Inhibitor VII；化合物 7a)是一种非肽、非竞争性和可逆的 caspase-3 抑制剂，IC50 为 23 nM，对其他胱天蛋白酶有一定选择性。

Emricasan（PF 03491390）是一种口服活性且不可逆的泛胱天蛋白酶抑制剂，可抑制寨卡病毒（ZIKV）引起的胱天蛋白酶-3活性增加并保护人类皮质神经祖细胞。

CASP3 Activator 1541 is an activator of procaspase-3.

Phytohemagglutinin (PHA-M), a lectin extract from the red kidney bean and a standard T cell mitogen, as an inhibitor of both T- and B-cell tumors. Phytohemagglutinin can inhibit incorporation of 3H-thymidine and mediate apoptosis of B- and T-cell tumor lines. Anti-tumor activity .

AS101 is a potent Caspase-1 inhibitor which can inhibit IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release through Caspase, performing as an immunomodulator.

Z-IETD-FMK is a specific Caspase-8 inhibitor.

Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate) prevents apoptosis by blocking a calcium-mediated apoptotic pathway as well as caspase-12 activation. Taurodeoxycholic acid sodium hydrate is investigated for use in several conditions such as Primary Biliary Cirrhosis (PBC), insulin resistance, amyloidosis, Cystic Fibrosis, Cholestasis, and Amyotrophic Lateral Sclerosis.

Z-DEVD-FMK (1–200 μM) inhibits D4-GDI cleavage and apoptosis in a concentration-dependent manner.

Aristolactam I是一种马兜铃酸I的主要代谢产物，直接作用于肾近端小管细胞，导致细胞毒性和肾损伤，其毒性效力高于AA-I，主要通过caspase-3依赖性细胞凋亡途径介导。

Dihydrocapsaicin, a natural product isolated and purified from the fruits of Capsicum annuum L..

AVN-944 is a selective, noncompetitive inhibitor of the enzyme directed against human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.

Yakuchinone A来源于 Alpinia oxyphylla，具有诱导细胞凋亡 (apoptosis)的活性，抗癌和抗炎的研究中显示出良好前景。

Ac-YVAD-cmk (Caspase-1 Inhibitor II) 是一种选择性的 caspase-1 (IL-1β 转化酶, ICE) 抑制剂，具有神经保护和抗炎作用。它有效抑制 IL-1β 和 IL-18 的表达，并在多种疾病中抑制细胞焦亡。

Senkyunolide I, a natural product isolated and purified from the roots of Ligusticum chuanxiong hort with anti-oxidation and anti-apoptosis properties, is traditionally used to treat migraine, can reduce the metamorphose damage of the RBC caused by ConA, alleviates the aggregation of the RBC, and protect rat brain against focal cerebral ischemia-reperfusion injury by up-regulating p-Erk1/2, Nrf2/HO-1 and inhibiting caspase 3.