BML-210 is the HDAC inhibitor, and its mechanism of action has not been characterized.

PF-3084014 is a reversible inhibitor of γ-secretase with IC50 of 6.2 nM.

NVS-CECR2-1 is a potent and selective CECR2 (cat eye syndrome chromosome region, candidate 2) inhibitor with IC50 of 47 nM.

T025是一种具有口服活性的 Cdc2-like 激酶 (CLK) 抑制剂，对多种 CLK 激酶亚型的 Kd 值在纳摩尔级别 (如 CLK2 为 0.096 nM)。T025 可诱导 caspase-3/7 介导的细胞凋亡，适用于 MYC 驱动的肿瘤和细胞增殖异常的疾病研究。

Casein Kinase inhibitor A86是一种有效且具有口服活性的酪蛋白激酶 1α (CK1α) 抑制剂，同时也抑制 CDK7 (TFIIH) 和 CDK9 (P-TEFb)，并能诱导白血病细胞凋亡 (apoptosis)，具有抗白血病活性。

Costunolide shows anti-inflammatory and anti-oxidant activities and also induces apoptosis. It is a sesquiterpene lactone isolated from stem bark of Magnolia sieboldii,

Inhibitor of checkpoint kinase 1 (Chk1) that displays selectivity over other protein kinases (IC50 values are 15, 250 and 1000 nM for Chk1, cdc2 and PKC respectively). Abrogates G2 cell cycle arrest caused by γ-irradiation and topoisomerase I inhibition. Potentiates cytotoxicity of DNA-damaging drugs, enhancing the efficacy of some chemotherapeutics.

PD184161 is an orally-active MEK inhibitor with antitumor effects in HCC in vitro and in vivo that appear to correlate with suppression of MEK activity.

Rilmenidine Phosphate is an oxazole-derived agonist of adrenergic receptor α2 and Imidazoline receptor, used in trials studying the treatment of hypertension and chronic kidney disease.

AOH1160是一种有效的、可口服的增殖细胞核抗原 (PCNA) 抑制剂，能够干扰 DNA 复制并阻断同源重组介导的 DNA 修复，进而导致细胞周期停滞并诱导细胞凋亡。AOH1160 适用于研究 DNA 损伤反应和癌症治疗中的潜在应用。

SSE15206 is a microtubule depolymerizing agent which inhibits microtubule polymerization both in biochemical and cellular assays by binding to colchicine site in tubulin. It causes aberrant mitosis resulting in G2/M arrest due to incomplete spindle formation.

LJH685 is a potent pan-RSK inhibitor with IC50 of 6 nM, 5 nM and 4 nM for RSK1, RSK2, and RSK3, respectively.

1A-116 is a specific Rac1 inhibitor.

Oncrasin-1 is a potent and effective anticancer inhibitor that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations and also leads to abnormal aggregation of PKCι in nucleus of sensitive cells but not in resistant cells.

Rotundifuran是一种从马鞭草属植物中分离的二萜类化合物，能通过抑制细胞周期进程并诱导凋亡，抑制骨髓性白血病细胞的增殖。

VER-50589 is an isoxazole compound that inhibits Hsp90 with an IC50 value of 21 nM.

Notopterol induces apoptosis and inhibits cell cycle-specific, it's a natural product isolated and purified from the roots of Notopterygium incisum.

QN523是一种新型化学骨架的分子，在 12 种癌细胞株中显示出强大的体外细胞毒性，能够诱导细胞凋亡 (apoptosis) 和自噬 (autophagy)，可用于癌症研究。

Baohuoside I, a flavonoid, acts as an apoptosis inducer and a down-regulator of durvivin and cyclin D1 expression. It is used as an anti-cancer agent and can be isolated and purified from the roots of epimedium brevicornu Maxim.

C-DIM12 is Nurr1 activator that stimulates Nurr1 mediated apoptosis axis in bladder cancer cells and tumors and inhibits NF-κB–dependent gene expression in glial cells.