| Hydroxyzine 2HCl |
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Cyclizine |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Loratadine |
+
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Desloratadine |
++
Histamine H1 receptor, IC50: 51 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Doxylamine succinate |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Ebastine |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Tripelennamine HCl |
+
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Meclizine dihydrochloride |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Chlorpheniramine maleate |
+++
Histamine H1 receptor, IC50: 12 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Diphenhydramine HCl |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Alcaftadine |
++++
|
++
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Fexofenadine HCl |
++
Histamine H1 receptor, IC50: 246 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Bilastine |
+++
H1 receptor, Ki: 44.15 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Pemirolast potassium |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Bepotastine besilate |
+
Histamine H1 receptor, pIC50: 5.7
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Mizolastine |
+++
Histamine H1 receptor, IC50: 47 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Brompheniramine maleate |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Carbinoxamine maleate salt |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Clemastine fumarate |
++++
Histamine H1 receptor, IC50: 3 nM
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Ketotifen fumarate salt |
✔
|
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Rupatadine Fumarate |
++
Histamine H1 receptor, Ki: 102 nM
|
|
|
|
|
PAFR
|
{[allProObj[0].p_purity_real_show]} |
| Famotidine |
|
✔
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Roxatidine Acetate HCl |
|
+
Histamine H2 receptor, IC50: 3.2 μM
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Lafutidine |
|
✔
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Cimetidine |
|
✔
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Nizatidine |
|
++++
Histamine H2 receptor, IC50: 0.9 nM
|
|
|
|
AChE
|
{[allProObj[0].p_purity_real_show]} |
| Ranitidine |
|
✔
|
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Betahistine |
|
|
+
Histamine H3 receptor, IC50: 1.9 μM
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Ciproxifan maleate |
|
|
+++
Histamine H3 receptor, IC50: 9.2 nM
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| S 38093 |
|
|
++
rat H3 receptor, Ki: 1.44 μM
human H3 receptor, Ki: 1.2 μM
|
|
|
|
{[allProObj[0].p_purity_real_show]} |
| JNJ-7777120 |
|
|
|
++++
Histamine H4 receptor, Ki: 4.5 nM
|
|
|
{[allProObj[0].p_purity_real_show]} |
| Azelastine HCl |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Epinastine HCl |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Levodropropizine |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Cyproheptadine hydrochloride |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Hesperetin |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Olopatadine HCl |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Mianserin hydrochloride |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Buclizine 2HCl |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
| Latrepirdine 2HCl |
|
|
|
|
✔
|
GluR
|
{[allProObj[0].p_purity_real_show]} |
| Cetirizine 2HCl |
|
|
|
|
✔
|
|
{[allProObj[0].p_purity_real_show]} |
|
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
|
搜索
