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G蛋白偶联受体/G蛋白
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/ 组胺受体 / Cyclizine

1-二苯甲基-4-甲基哌嗪 /Cyclizine {[allProObj[0].p_purity_real_show]}

货号：A348582

Cyclizine, a piperazine derivative, is an antihistaminic antiemetic that is useful in the prevention and treatment of nausea and vomiting associated with motion sickness.

HazMat Fee +

There will be a HazMat fee per item when shipping a dangerous goods. The HazMat fee will be charged to your UPS/DHL/FedEx collect account or added to the invoice unless the package is shipped via Ground service. Ship by air in Excepted Quantity (each bottle), which is up to 1g/1mL for class 6.1 packing group I or II, and up to 25g/25ml for all other HazMat items.

Type HazMat fee for 500 gram (Estimated)
Excepted Quantity USD 0.00
Limited Quantity USD 15-60
Inaccessible (Haz class 6.1), Domestic USD 80+
Inaccessible (Haz class 6.1), International USD 150+
Accessible (Haz class 3, 4, 5 or 8), Domestic USD 100+
Accessible (Haz class 3, 4, 5 or 8), International USD 200+
Cyclizine 化学结构 CAS号：82-92-8
Cyclizine 化学结构
CAS号：82-92-8
Cyclizine 3D分子结构
CAS号：82-92-8
Cyclizine 化学结构 CAS号：82-92-8
Cyclizine 3D分子结构 CAS号：82-92-8
规格 价格 会员价 库存 数量
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Cyclizine 纯度/质量文件 产品仅供科研

货号：A348582 标准纯度： {[allProObj[0].p_purity_real_show]}
批次查询： 批次纯度:

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产品名称 H1 receptor ↓ H2 receptor ↓ H3 receptor ↓ H4 receptor ↓ Histamine receptor ↓ 其他靶点 纯度
Hydroxyzine 2HCl 99+%
Cyclizine ✔ 97%
Loratadine +

B(0)AT2, IC50: 4 μM

 		98%
Desloratadine ++

Histamine H1 receptor, IC50: 51 nM

 		98%
Doxylamine succinate ✔ 99%
Ebastine ✔ 98%
Tripelennamine HCl +

H1 receptor, IC50: 30 μM

 		98%
Meclizine dihydrochloride ✔ 98%
Chlorpheniramine maleate +++

Histamine H1 receptor, IC50: 12 nM

 		99%
Diphenhydramine HCl ✔ 99%
Alcaftadine ++++

H1 receptor, pKi: 8.5

 		++

H2 receptor, pKi: 7.2

 		99%+
Fexofenadine HCl ++

Histamine H1 receptor, IC50: 246 nM

 		99%+
Bilastine +++

H1 receptor, Ki: 44.15 nM

 		98%
Pemirolast potassium ✔ 98%
Bepotastine besilate +

Histamine H1 receptor, pIC50: 5.7

 		98%
Mizolastine +++

Histamine H1 receptor, IC50: 47 nM

 		98%
Brompheniramine maleate ✔ 98%
Carbinoxamine maleate salt ✔ 99+%
Clemastine fumarate ++++

Histamine H1 receptor, IC50: 3 nM

 		98%
Ketotifen fumarate salt ✔ 95%
Rupatadine Fumarate ++

Histamine H1 receptor, Ki: 102 nM

 		PAFR 98%
Famotidine ✔ 97%
Roxatidine Acetate HCl +

Histamine H2 receptor, IC50: 3.2 μM

 		98%
Lafutidine ✔ 99%
Cimetidine ✔ 98%
Nizatidine ++++

Histamine H2 receptor, IC50: 0.9 nM

 		AChE 98%
Ranitidine ✔ 99%
Betahistine +

Histamine H3 receptor, IC50: 1.9 μM

 		98%
Ciproxifan maleate +++

Histamine H3 receptor, IC50: 9.2 nM

 		99%+
S 38093 ++

rat H3 receptor, Ki: 1.44 μM

human H3 receptor, Ki: 1.2 μM

 		98%
JNJ-7777120 ++++

Histamine H4 receptor, Ki: 4.5 nM

 		98%
Azelastine HCl ✔ 98%
Epinastine HCl ✔ 98%
Levodropropizine ✔ 97%
Cyproheptadine hydrochloride ✔ 98%
Hesperetin ✔ 97%
Olopatadine HCl ✔ 98%
Mianserin hydrochloride ✔ 99+%
Buclizine 2HCl ✔ 97%
Latrepirdine 2HCl ✔ GluR 98%
Cetirizine 2HCl ✔ 98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。

Cyclizine 生物活性

靶点

  • H1 receptor
描述 Cyclizine, a piperazine derivative, is an antihistaminic antiemetic that is useful in the prevention and treatment of nausea and vomiting associated with motion sickness.

Cyclizine 临床研究

NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点
NCT01303809 Morbid Obesity Not Applicable Completed - New Zealand ... 展开 >> Manukau Surgery Centre Auckland, New Zealand, 2025 收起 <<
NCT02009306 Terminal Cancer Phase 4 Completed - United Kingdom ... 展开 >> Sue Ryder Leckhampton Court Hospice Cheltenham, Gloucestershire, United Kingdom, GL53 0QJ 收起 <<
NCT02288923 Arthritis Knee Not Applicable Recruiting April 30, 2018 United Kingdom ... 展开 >> Royal Devon and Exeter NHS Foundation Trust Recruiting Exeter, Devon, United Kingdom, EX2 5DW Contact: Fiona Martin, MBCHB    +441392411611 ext 2474    fiona.martin8@nhs.net    Sub-Investigator: James Cockcroft, MBCHB          Sub-Investigator: James Simpson, MBCHB 收起 <<

Cyclizine 实验方案

计算器
存储液制备 1mg 5mg 10mg

1 mM

5 mM

10 mM

3.75mL

0.75mL

0.38mL

18.77mL

3.75mL

1.88mL

37.54mL

7.51mL

3.75mL

Cyclizine 技术信息

CAS号82-92-8
分子式C18H22N2
分子量 266.381
别名
运输蓝冰
存储条件

液体 -20°C:3-6个月-80°C:12个月

粉末 Sealed in dry,Room Temperature
溶解度

DMSO: 105 mg/mL(394.17 mM)，配合低频超声助溶，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO
动物实验配方

Tags: Cyclizine | Histamine Receptor | AmBeed-信号通路专用抑制剂 | Cyclizine 纯度/质量文件 | Cyclizine 亚型比较 | Cyclizine 生物活性 | Cyclizine 临床数据 | Cyclizine 实验方案 | Cyclizine 技术信息

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