GSK189254A
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货号：A884075
同义名：
GSK189254
GSK189254A 是一种强效且选择性的组胺 H3 受体拮抗剂，人类和大鼠 H3 受体的 pKi 值分别为 9.59-9.90 和 8.51-9.17。
GSK189254A 化学结构
CAS号：720690-73-3
GSK189254A 3D分子结构
CAS号：720690-73-3
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GSK189254A 纯度/质量文件 产品仅供科研
货号：A884075
标准纯度：
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GSK189254A 质控信息
| Hydroxyzine 2HCl |
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99+% |
| Cyclizine |
✔
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97% |
| Loratadine |
+
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98% |
| Desloratadine |
++
Histamine H1 receptor, IC50: 51 nM
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98% |
| Doxylamine succinate |
✔
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99% |
| Ebastine |
✔
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98% |
| Tripelennamine HCl |
+
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98% |
| Meclizine dihydrochloride |
✔
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98% |
| Chlorpheniramine maleate |
+++
Histamine H1 receptor, IC50: 12 nM
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99% |
| Diphenhydramine HCl |
✔
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99% |
| Alcaftadine |
++++
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++
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99%+ |
| Fexofenadine HCl |
++
Histamine H1 receptor, IC50: 246 nM
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99%+ |
| Bilastine |
+++
H1 receptor, Ki: 44.15 nM
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98% |
| Pemirolast potassium |
✔
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98% |
| Bepotastine besilate |
+
Histamine H1 receptor, pIC50: 5.7
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98% |
| Mizolastine |
+++
Histamine H1 receptor, IC50: 47 nM
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98% |
| Brompheniramine maleate |
✔
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98% |
| Carbinoxamine maleate salt |
✔
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99+% |
| Clemastine fumarate |
++++
Histamine H1 receptor, IC50: 3 nM
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98% |
| Ketotifen fumarate salt |
✔
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95% |
| Rupatadine Fumarate |
++
Histamine H1 receptor, Ki: 102 nM
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PAFR
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98% |
| Famotidine |
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✔
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97% |
| Roxatidine Acetate HCl |
|
+
Histamine H2 receptor, IC50: 3.2 μM
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98% |
| Lafutidine |
|
✔
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99% |
| Cimetidine |
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✔
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98% |
| Nizatidine |
|
++++
Histamine H2 receptor, IC50: 0.9 nM
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AChE
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98% |
| Ranitidine |
|
✔
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98% |
| Betahistine |
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|
+
Histamine H3 receptor, IC50: 1.9 μM
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98% |
| Ciproxifan maleate |
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+++
Histamine H3 receptor, IC50: 9.2 nM
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99%+ |
| S 38093 |
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++
human H3 receptor, Ki: 1.2 μM
rat H3 receptor, Ki: 1.44 μM
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98% |
| JNJ-7777120 |
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++++
Histamine H4 receptor, Ki: 4.5 nM
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98% |
| Azelastine HCl |
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✔
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98% |
| Epinastine HCl |
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✔
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98% |
| Levodropropizine |
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✔
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97% |
| Cyproheptadine hydrochloride |
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✔
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98% |
| Hesperetin |
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✔
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97% |
| Olopatadine HCl |
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✔
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98% |
| Mianserin hydrochloride |
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✔
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99+% |
| Buclizine 2HCl |
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✔
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97% |
| Latrepirdine 2HCl |
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✔
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GluR
|
98% |
| Cetirizine 2HCl |
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✔
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98% |
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1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
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GSK189254A 生物活性
| 描述 |
GSK189254A is a potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. |
GSK189254A 参考文献
GSK189254A 实验方案
| 计算器 |
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| 存储液制备 |
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1mg |
5mg |
10mg |
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1 mM
5 mM
10 mM
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2.85mL
0.57mL
0.28mL
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14.23mL
2.85mL
1.42mL
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28.45mL
5.69mL
2.85mL
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GSK189254A 技术信息
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