Ambeed.cn

首页 / 抑制剂/激动剂 / 代谢酶 / 碳酸酐酶

货号 产品名 纯度
A554211 现货 2-Aminobenzenesulfonamide/2-氨基苯磺酰胺

2-Aminobenzenesulfonamide is a potent inhibitor of carbonic anhydrase B.

98%
A1258800 现货 CAIX Inhibitor S4

S4 is a selective inhibitor of CA IX and CA XII inhibitor. The Ki values are 2, 7, 547 and 5600 nM for CA XII, IX, II and I, respectively.

99%+
A1868758 现货 hCAII-IN-8

hCAII-IN-8是一种酰胺类化合物,是一种高选择性的碳酸酐酶 (CA) 抑制剂,对 hCA II 的 IC50 为 0.18 μM。

99%+
A876758 现货 Ethoxzolamide/依索唑胺

Ethoxzolamide is an inhibitor of carbonic anhydrase with (Ki = 1 nM).

99%+
A906540 现货 Benzolamide

Benzolamide是一种有效的碳酸酐酶 (CA) 抑制剂,能够抑制多种碳酸酐酶亚型 (hCA I、hCA II、EcoCAγ、VchCAγ和CAS3),适用于青光眼和癫痫的研究,并展示了在这些疾病中的治疗潜力。

99%+
A407281 现货 Methyclothiazide/甲氯噻嗪

Methyclothiazide is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions including heart disease.

98%
A580496 现货 Polmacoxib

Polmacoxib是一种双重抑制剂,抑制 COX-2 (IC50 ~ 0.1 μg/ml) 和碳酸酐酶,具有口服活性。该药物在小鼠模型中表现出抑制大肠腺瘤和肿瘤生长的能力,具有抗炎抗肿瘤潜力,适用于癌症及炎症疾病的研究。

97%
A275314 现货 Mafenide HCl/盐酸磺胺米隆

Mafenide HCl is a sulfonamide that inhibits the enzyme carbonic anhydrase and is used as a topical anti-bacterial agent, especially in burn therapy.

98%
A119509 现货 Benzenesulphonamide/苯磺酰胺

Benzenesulfonamide ia an inhibitor of carbonic anhydrases.

98%
A1678235 现货 hCAI/II-IN-6

hCAI/II-IN-6是一种口服活性的碳酸酐酶 (CA) 抑制剂,具有选择性,尤其对 hCA II 和 hCA VII 显示较强抑制活性,主要用于癫痫及抗惊厥药物的研究。

99%+
A1417612 现货 EMAC10101d

EMAC10101d is a potent and selective Carbonic Anhydrase II inhibitor.

99%+
A637802 现货 Sultiame/舒噻嗪

Sultiame is an inhibitor of carbonic anhydrase that used to treat epilepsy.

99%+
A436967 现货 Tioxolone/噻克索酮

Tioxolone, a metalloenzyme carbonic anhydrase I inhibitor with a Ki of 91 nM, is an anti-acne preparation.

98%
A112487 现货 U-104

U-104 is a potent carbonic anhydrase (CA) inhibitor with Ki of 45.1 nM and 4.5 nM for CA IX and CA XII, respectively.

98%
A615855 现货 Dimethylfraxetin

Dimethylfraxetin is a natural product isolated and purified from the herbs of Viola yedonensis Makino with anti-HRV-2 activity.

98%
A201176 现货 Dichlorphenamide/二氯苯二磺胺

Dichlorphenamide is a sulfonamide and an orally bioavailable carbonic anhydrase (CA) inhibitor with Kis of 1.20, 38, 50, and 50 nM for the human CA isoforms CAI, CAII, CAIX, and CAXII, respectively.

98%
A730578 现货 Diclazuril/地克珠利

Diclazuril is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.

98%
A160451 现货 Methocarbamol/美索巴莫

Methocarbamol is a central muscle relaxant used to treat skeletal muscle spasms.

98%
A120295 现货 Methazolamide/醋甲唑胺

Methazolamide is a carbonic anhydrase inhibitor with Ki of 50 nM, 14 nM and 36 nM for hCA I, hCA II and bCA IV isoforms, respectively.

98%
A525496 现货 Dorzolamide HCl/盐酸多佐胺

Dorzolomide HCl is a potent and water-soluble inhibitor of human carbonic anhydrase II and IV with Ki of 1.9 nM and 31 nM respectively and used as anti-glaucoma agent.

98%
产品名 Carbonic Anhydrase Carbonic Anhydrase I Carbonic Anhydrase II Carbonic Anhydrase IV Carbonic Anhydrase IX Carbonic Anhydrase XII 其他靶点 纯度
Topiramate Calcium Channel 98%
Dichlorphenamide 98%
Mafenide Acetate 98%
Benzenesulphonamide 98%
Dorzolamide HCl +

Carbonic anhydrase I, Ki: 6000 nM

++++

Carbonic anhydrase II, Ki: 1.9 nM

+++

Carbonic anhydrase IV, Ki: 31 nM

98%
Methazolamide ++

hCAI, Ki: 50 nM

+++

hCAII, Ki: 14 nM

++

bCAIV, Ki: 36 nM

98%
Tioxolone +

CAI, Ki: 91 nM

98%
U-104 ++

CAIX, Ki: 45.1 nM

++++

CAXII, Ki: 4.5 nM

98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
Ambeed 相关网站 Ambeed.cn Ambeed.com
Ambeed
关于我们
联系我们
资讯中心
网站地图
产品手册
  • 批次文件查询
  • 客户支持
    技术支持
    专业术语
    缩略词释义
    质量手册
    产品咨询
    计算器
    活动政策
    订购方法
    积分商城
    活动声明
    联系我们
    400-920-2911 sales@ambeed.cn tech@ambeed.cn
    Ambeed 只为有资质的科研机构、医药企业基于科学研究或药证申报的用途提供医药研发服务,不为任何个人或者非科研性质用途提供服务。