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AG-825 {[allProObj[0].p_purity_real_show]}

货号:A276278 同义名: Tyrphostin AG-825 Ambeed 开学季,买赠积分,赢豪礼

AG-825 是一种选择性、ATP竞争性的ErbB2酪氨酸磷酸化抑制剂,IC50值为0.35 μM。AG-825具有抗癌活性,并显著加速人类中性粒细胞的凋亡。它在克服锰诱导的神经毒性或阿尔茨海默病发展中是一种潜在的活性分子。

AG-825 化学结构 CAS号:149092-50-2
AG-825 化学结构
CAS号:149092-50-2
AG-825 3D分子结构
CAS号:149092-50-2
AG-825 化学结构 CAS号:149092-50-2
AG-825 3D分子结构 CAS号:149092-50-2
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AG-825 纯度/质量文件 产品仅供科研

货号:A276278 标准纯度: {[allProObj[0].p_purity_real_show]}
批次查询: 批次纯度:

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产品名称 Cdc CDK1 CDK19 CDK2 CDK3 CDK4 CDK5 CDK6 CDK7 CDK8 CDK9 CLK 其他靶点 纯度
XL413 hydrochloride ++++

Cdc7, IC50: 3.4 nM

{[allProObj[0].p_purity_real_show]}
SU9516 +++

CDK1, IC50: 40 nM

+++

CDK2, IC50: 22 nM

++

CDK4, IC50: 200 nM

{[allProObj[0].p_purity_real_show]}
RO-3306 +++

CDK1, Ki: 20 nM

ERK,SGK {[allProObj[0].p_purity_real_show]}
R547 ++++

CDK1/CyclinB, Ki: 2 nM

++++

CDK2/CyclinE, Ki: 3 nM

++++

CDK4/CyclinD1, Ki: 1 nM

{[allProObj[0].p_purity_real_show]}
BMS-265246 ++++

CDK1/CyclinB, IC50: 6 nM

++++

CDK2/CyclinE, IC50: 9 nM

+

CDK4/CyclinD, IC50: 230 nM

{[allProObj[0].p_purity_real_show]}
NU6027 +

CDK1, Ki: 2.5 μM

+

CDK2, Ki: 1.3 μM

DNA-PK {[allProObj[0].p_purity_real_show]}
Purvalanol A ++++

Cdc2/CyclinB, IC50: 4 nM

+++

CDK2/CyclinE, IC50: 35 nM

CDK2/CyclinA, IC50: 70 nM

+

CDK4/CyclinD1, IC50: 850 nM

{[allProObj[0].p_purity_real_show]}
SCH900776 ++

CDK2, IC50: 0.16 μM

{[allProObj[0].p_purity_real_show]}
AUZ 454 ++++

CDK2(C118L), Kd: 18.6 nM

CDK2(A144C), Kd: 9.7 nM

{[allProObj[0].p_purity_real_show]}
A-674563 HCl ++

CDK2, Ki: 46 nM

PKA {[allProObj[0].p_purity_real_show]}
JNJ-7706621 ++++

CDK1/CyclinB, IC50: 9 nM

++++

CDK2/CyclinE, IC50: 3 nM

CDK2/CyclinA, IC50: 4 nM

++

CDK3/CyclinE, IC50: 58 nM

+

CDK4/CyclinD1, IC50: 253 nM

++

CDK6/CyclinD1, IC50: 175 nM

{[allProObj[0].p_purity_real_show]}
AT7519 ++

CDK1/CyclinB, IC50: 210 nM

++

CDK2/CyclinA, IC50: 47 nM

+

CDK3/CyclinE, IC50: 360 nM

++

CDK4/CyclinD1, IC50: 100 nM

+++

CDK5/p35, IC50: 13 nM

++

CDK6/CyclinD3, IC50: 170 nM

++++

CDK9/CyclinT, IC50: <10 nM

{[allProObj[0].p_purity_real_show]}
PHA-793887 ++

CDK1/CyclinB, IC50: 60 nM

++++

CDK2/CyclinE, IC50: 8 nM

CDK2/CyclinA, IC50: 8 nM

++

CDK4/CyclinD1, IC50: 62 nM

++++

CDK5/p25, IC50: 5 nM

++++

CDK7/CyclinH, IC50: 10 nM

++

CDK9/CyclinT1, IC50: 138 nM

{[allProObj[0].p_purity_real_show]}
Milciclib +

CDK1/CyclinB, IC50: 398 nM

++

CDK2/CyclinE, IC50: 363 nM

CDK2/CyclinA, IC50: 45 nM

++

CDK4/CyclinD1, IC50: 160 nM

+

CDK5/p35, IC50: 265 nM

++

CDK7/CyclinH, IC50: 150 nM

{[allProObj[0].p_purity_real_show]}
Kenpaullone +

CDK1/CyclinB, IC50: 0.4μM

+

CDK2/CyclinE, IC50: 7.5μM

CDK2/CyclinA, IC50: 0.68μM

+

CDK5/p35, IC50: 0.85μM

{[allProObj[0].p_purity_real_show]}
SNS-032 +++

CDK2/CyclinE, IC50: 48 nM

CDK2/CyclinA, IC50: 38 nM

+

CDK5/p35, IC50: 340 nM

++

CDK7/CyclinH, IC50: 62 nM

++++

CDK9/CyclinT, IC50: 4 nM

{[allProObj[0].p_purity_real_show]}
Dinaciclib ++++

CDK1, IC50: 3 nM

++++

CDK2, IC50: 1 nM

++++

CDK5, IC50: 1 nM

++++

CDK9, IC50: 4 nM

{[allProObj[0].p_purity_real_show]}
PHA-767491 hydrochloride ++++

Cdc7, IC50: 10 nM

+

CDK1, IC50: 250 nM

+

CDK2, IC50: 240 nM

+

CDK5, IC50: 460 nM

+++

CDK9, IC50: 34 nM

MK2 {[allProObj[0].p_purity_real_show]}
(R)-Roscovitine +

Cdc2/CyclinB, IC50: 0.65 μM

+

CDK2/CyclinE, IC50: 0.7 μM

CDK2/CyclinA, IC50: 0.7 μM

++

CDK5/p35, IC50: 0.16 μM

{[allProObj[0].p_purity_real_show]}
Narazaciclib ++++

CDK4/CyclinD1, IC50: 3.87 nM

++++

CDK6/CyclinD1, IC50: 9.82 nM

RET {[allProObj[0].p_purity_real_show]}
Palbociclib ++++

CDK4/CyclinD1, IC50: 11 nM

CDK4/CyclinD3, IC50: 9 nM

+++

CDK6/CyclinD2, IC50: 15 nM

{[allProObj[0].p_purity_real_show]}
Abemaciclib ++++

CDK4, IC50: 2 nM

++++

CDK6, IC50: 10 nM

{[allProObj[0].p_purity_real_show]}
Ribociclib ++++

CDK4, IC50: 10 nM

+++

CDK6, IC50: 39 nM

{[allProObj[0].p_purity_real_show]}
Palbociclib isethionate ++++

CDK4/CyclinD1, IC50: 11 nM

CDK4/CyclinD3, IC50: 9 nM

+++

CDK6/CyclinD2, IC50: 15 nM

{[allProObj[0].p_purity_real_show]}
BS-181 HCl +++

CDK7, IC50: 21 nM

{[allProObj[0].p_purity_real_show]}
(E/Z)-THZ1 dihydrochloride ++++

CDK7, IC50: 3.2 nM

{[allProObj[0].p_purity_real_show]}
LDC4297 ++++

CDK7, IC50: 0.13 nM

{[allProObj[0].p_purity_real_show]}
Senexin A +

CDK19, Kd: 0.31 μM

+

CDK8, Kd: 0.83 μM

{[allProObj[0].p_purity_real_show]}
MSC2530818 ++++

CDK8, IC50: 2.6 nM

{[allProObj[0].p_purity_real_show]}
Wogonin {[allProObj[0].p_purity_real_show]}
Riviciclib HCl ++

CDK1/CyclinB, IC50: 79 nM

+

CDK2/CyclinE, IC50: 2.54 μM

CDK2/CyclinA, IC50: 224 nM

++

CDK4/CyclinD1, IC50: 63 nM

+

CDK6/CyclinD3, IC50: 396 nM

+

CDK7/CyclinH, IC50: 2.87 μM

+++

CDK9/CyclinT1, IC50: 20 nM

{[allProObj[0].p_purity_real_show]}
LDC000067 +

CDK2, IC50: 2.441 μM

++

CDK9, IC50: 44 nM

{[allProObj[0].p_purity_real_show]}
Flavopiridol +++

CDK1, IC50: 40 nM

+++

CDK2, IC50: 40 nM

+++

CDK4, IC50: 40 nM

+++

CDK6, IC50: 40 nM

+

CDK7, IC50: 300 nM

+++

CDK9, IC50: 20 nM

{[allProObj[0].p_purity_real_show]}
LY2857785 +

CDK7, IC50: 0.246 μM

+++

CDK8, IC50: 0.016 μM

+++

CDK9, IC50: 0.011 μM

{[allProObj[0].p_purity_real_show]}
AZD-5438 +++

CDK1, IC50: 16 nM

++++

CDK2, IC50: 6 nM

+++

CDK9, IC50: 20 nM

{[allProObj[0].p_purity_real_show]}
ML167 ++

Dyrk1B , IC50: 1648 nM

CLK4, IC50: 136 nM

{[allProObj[0].p_purity_real_show]}
(E/Z)-TG003 +++

mCLK1, IC50: 200 nM

mCLK4, IC50: 15 nM

{[allProObj[0].p_purity_real_show]}
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
产品名称 EGFR/ErbB1 ErbB3 ErbB4 HER2/ErbB2 mutant EGFR 其他靶点 纯度
WZ-3146 ++++

EGFR (E746_A750/T790M), IC50: 14 nM

EGFR (E746_A750), IC50: 2 nM

{[allProObj[0].p_purity_real_show]}
Daphnetin +

EGFR, IC50: 7.67 μM

PKA,PKC {[allProObj[0].p_purity_real_show]}
Lifirafenib ++

EGFR, IC50: 29 nM

+

EGFR(T790M/L858R), IC50: 495 nM

{[allProObj[0].p_purity_real_show]}
PD168393 ++++

EGFR, IC50: 0.70 nM

{[allProObj[0].p_purity_real_show]}
Nazartinib ++

mutant EGFR, Ki: 0.031 μM

++

mutant EGFR, Ki: 0.031 μM

{[allProObj[0].p_purity_real_show]}
Norcantharidin {[allProObj[0].p_purity_real_show]}
CL-387785 ++++

EGFR, IC50: 370 pM

{[allProObj[0].p_purity_real_show]}
WHI-P154 +++

EGFR, IC50: 4 nM

VEGFR,Src {[allProObj[0].p_purity_real_show]}
Tyrphostin A9 +

EGFR, IC50: 460 μM

PDGFR {[allProObj[0].p_purity_real_show]}
AG 555 +

EGFR, IC50: 0.7 μM

{[allProObj[0].p_purity_real_show]}
AG 494 +

EGFR, IC50: 1.2 μM

{[allProObj[0].p_purity_real_show]}
AG-556 +

EGFR, IC50: 5 μM

{[allProObj[0].p_purity_real_show]}
RG13022 +

EGFR, IC50: 4 μM

{[allProObj[0].p_purity_real_show]}
Tyrphostin RG 14620 {[allProObj[0].p_purity_real_show]}
Vandetanib +

EGFR, IC50: 500 nM

{[allProObj[0].p_purity_real_show]}
CNX-2006 ++

mutant EGFR, IC50: <20 nM

++

mutant EGFR, IC50: <20 nM

{[allProObj[0].p_purity_real_show]}
AZD3759 ++++

EGFR (WT), IC50: 0.3 nM

EGFR (L858R), IC50: 0.2 nM

{[allProObj[0].p_purity_real_show]}
Erlotinib ++++

EGFR, IC50: 2 nM

{[allProObj[0].p_purity_real_show]}
Saracatinib +++

EGFR, IC50: 5 nM

EGFR (L861Q), IC50: 4 nM

{[allProObj[0].p_purity_real_show]}
AG1557 {[allProObj[0].p_purity_real_show]}
Rociletinib ++

EGFR (L858R/T790M), Ki: 21.5 nM

EGFR (wt), Ki: 303.3 nM

{[allProObj[0].p_purity_real_show]}
AG490 +

EGFR, IC50: 0.1 μM

{[allProObj[0].p_purity_real_show]}
Cetuximab ++++

EGFR, Kd: 0.39 nM

{[allProObj[0].p_purity_real_show]}
Osimertinib ++

L858R/T790M EGFR, IC50: 11.44 nM

WT EGFR, IC50: 12.92 nM

{[allProObj[0].p_purity_real_show]}
Osimertinib mesylate {[allProObj[0].p_purity_real_show]}
Chrysophanol mTOR {[allProObj[0].p_purity_real_show]}
PD153035 ++++

EGFR, Ki: 5.2 pM

{[allProObj[0].p_purity_real_show]}
Olmutinib BTK {[allProObj[0].p_purity_real_show]}
WZ4002 ++++

EGFR (L858R/T790M), IC50: 8 nM

EGFR (L858R), IC50: 2 nM

{[allProObj[0].p_purity_real_show]}
Icotinib +++

EGFR, IC50: 5 nM

{[allProObj[0].p_purity_real_show]}
Desmethyl Erlotinib HCl ++++

EGFR, IC50: 2 nM

{[allProObj[0].p_purity_real_show]}
Cyasterone {[allProObj[0].p_purity_real_show]}
PP 3 +

EGFR tyrosine kinase, IC50: 2.7 μM

{[allProObj[0].p_purity_real_show]}
WZ8040 {[allProObj[0].p_purity_real_show]}
(-)-Epigallocatechin Gallate {[allProObj[0].p_purity_real_show]}
AG 18 +

EGFR, IC50: 35 μM

{[allProObj[0].p_purity_real_show]}
O-Desmethyl gefitinib ++

EGFR, IC50: 36 nM

{[allProObj[0].p_purity_real_show]}
Falnidamol {[allProObj[0].p_purity_real_show]}
AZ-5104 ++++

EGFR (L858R), IC50: 6 nM

EGFR (L861Q) , IC50: <1 nM

+++

ErbB4, IC50: 7 nM

BRK {[allProObj[0].p_purity_real_show]}
Butein {[allProObj[0].p_purity_real_show]}
Genistein {[allProObj[0].p_purity_real_show]}
SU5214 +

EGFR, IC50: 36.7 μM

{[allProObj[0].p_purity_real_show]}
Naquotinib {[allProObj[0].p_purity_real_show]}
Gefitinib ++

EGFR, IC50: 15.5 nM

+

EGFR (858R/T790M), IC50: 823.3 nM

{[allProObj[0].p_purity_real_show]}
Theliatinib +++

WT EGFR, IC50: 3 nM

++

EGFR T790M/L858R, IC50: 22 nM

{[allProObj[0].p_purity_real_show]}
Lazertinib ++++

L858R/T790M EGFR, IC50: 2 nM

WT EGFR, IC50: 76 nM

++++

Del19/T790M, IC50: 1.7 nM

{[allProObj[0].p_purity_real_show]}
Gefitinib-based PROTAC 3 ++

EGFR, DC50: 22.3 nM

{[allProObj[0].p_purity_real_show]}
MTX-211 PI3K {[allProObj[0].p_purity_real_show]}
(E)-AG 99 {[allProObj[0].p_purity_real_show]}
Licochalcone D PARP,Caspase {[allProObj[0].p_purity_real_show]}
Zipalertinib +++

EGFR WT, IC50: 8 nM

EGFR (L861Q), IC50: 4.1 nM

+++

HER4, IC50: 4 nM

++++

EGFR L858R, IC50: 2 nM

EGFR(d746-750), IC50: 1.4 nM

{[allProObj[0].p_purity_real_show]}
JND3229 +++

EGFR WT, IC50: 6.8 nM

++

EGFR L858R/T790M, IC50: 30.5 nM

{[allProObj[0].p_purity_real_show]}
Firmonertinib mesylate {[allProObj[0].p_purity_real_show]}
Tyrphostin AG30 {[allProObj[0].p_purity_real_show]}
EGFR-IN-12 ++

EGFR, IC50: 21 nM

{[allProObj[0].p_purity_real_show]}
Mobocertinib {[allProObj[0].p_purity_real_show]}
(Rac)-JBJ-04-125-02 {[allProObj[0].p_purity_real_show]}
(S)-Sunvozertinib {[allProObj[0].p_purity_real_show]}
BLU-945 {[allProObj[0].p_purity_real_show]}
Poziotinib +++

HER1, IC50: 3.2 nM

++

HER4, IC50: 23.5 nM

+++

HER2, IC50: 5.3 nM

{[allProObj[0].p_purity_real_show]}
TAK-285 ++

EGFR/HER1, IC50: 23 nM

+

HER4, IC50: 260 nM

++

HER2, IC50: 17 nM

{[allProObj[0].p_purity_real_show]}
ARRY-380 analog {[allProObj[0].p_purity_real_show]}
Canertinib ++++

EGFR, IC50: 1.5 nM

+++

ErbB2, IC50: 9.0 nM

{[allProObj[0].p_purity_real_show]}
Dacomitinib +++

EGFR, IC50: 6.0 nM

+

ErbB4, IC50: 73.7 nM

+

ErbB2, IC50: 45.7 nM

{[allProObj[0].p_purity_real_show]}
EGFR/ErbB-2/ErbB-4 inhibitor-2 +

ErbB4, IC50: 1.91 μM

+

ErbB2, IC50: 0.08 μM

{[allProObj[0].p_purity_real_show]}
(E/Z)-CP-724714 ++

HER2/ErbB2, IC50: 10 nM

{[allProObj[0].p_purity_real_show]}
Lapatinib ++

EGFR, IC50: 10.8 nM

+

ErbB4, IC50: 367 nM

+++

ErbB2, IC50: 9.2 nM

{[allProObj[0].p_purity_real_show]}
AEE788 ++++

EGFR, IC50: 2 nM

+

HER4/ErbB4, IC50: 160 nM

+++

HER2/ErbB2, IC50: 6 nM

c-Fms {[allProObj[0].p_purity_real_show]}
AV-412 free base ++++

EGFR, IC50: 0.75 nM

++

ErbB2, IC50: 19 nM

++++

EGFRT790M, IC50: 0.79 nM

EGFRL858R/T790M, IC50: 0.51 nM

{[allProObj[0].p_purity_real_show]}
Neratinib +

EGFR, IC50: 92 nM

+

HER2, IC50: 59 nM

Src {[allProObj[0].p_purity_real_show]}
BMS-599626 ++

HER1, IC50: 20 nM

+

HER4, IC50: 190 nM

++

HER2, IC50: 30 nM

{[allProObj[0].p_purity_real_show]}
Tucatinib +++

ErbB2, IC50: 8 nM

{[allProObj[0].p_purity_real_show]}
Allitinib ++++

EGFR, IC50: 0.5 nM

++++

ErbB4, IC50: 0.8 nM

+++

ErbB2, IC50: 3.0 nM

{[allProObj[0].p_purity_real_show]}
Pelitinib +

EGFR, IC50: 38.5 nM

+

ErbB2, IC50: 1.255 μM

Raf,Src {[allProObj[0].p_purity_real_show]}
Sapitinib +++

EGFR, IC50: 4 nM

+++

ErbB3, IC50: 4 nM

+++

ErbB2, IC50: 3 nM

{[allProObj[0].p_purity_real_show]}
CUDC-101 +++

EGFR, IC50: 2.4 nM

++

HER2, IC50: 15.7 nM

HDAC {[allProObj[0].p_purity_real_show]}
Varlitinib +++

ErbB1, IC50: 7 nM

++++

ErbB2, IC50: 2 nM

{[allProObj[0].p_purity_real_show]}
Afatinib dimaleate ++++

EGFR (L858R/T790M), IC50: 0.4 nM

EGFR (wt), IC50: 0.5 nM

++

HER2, IC50: 14 nM

{[allProObj[0].p_purity_real_show]}
Canertinib dihydrochloride +++

EGFR, IC50: 7.4 nM

+++

ErbB2, IC50: 9 nM

{[allProObj[0].p_purity_real_show]}
Allitinib tosylate ++++

EGFR (T790M/L858R), IC50: 12 nM

EGFR, IC50: 0.5 nM

++++

ErbB4, IC50: 0.8 nM

+++

ErbB2, IC50: 3.0 nM

{[allProObj[0].p_purity_real_show]}
Tyrphostin AG 528 +

EGFR, IC50: 4.9 μM

+

HER2, IC50: 2.1 μM

{[allProObj[0].p_purity_real_show]}
Afatinib ++++

EGFR (L858R), IC50: 10 nM

EGFR (wt), IC50: 0.5 nM

++++

ErbB4, IC50: 1 nM

++

HER2, IC50: 14 nM

{[allProObj[0].p_purity_real_show]}
Pyrotinib dimaleate ++

EGFR, IC50: 0.013 μM

++

HER2, IC50: 0.038 μM

{[allProObj[0].p_purity_real_show]}
Epertinib HCl ++++

EGFR, IC50: 1.48 nM

+++

HER4, IC50: 2.49 nM

+++

HER2, IC50: 7.15 nM

{[allProObj[0].p_purity_real_show]}
Tuxobertinib ++++

EGFR, Kd: 0.2 nM

++++

HER2, Kd: 0.76 nM

{[allProObj[0].p_purity_real_show]}
ALK-IN-1 ++

EGFR(C797S/del19), IC50: 138.6 nM

EGFR(del19), IC50: 36.8 nM

ALK {[allProObj[0].p_purity_real_show]}
Brigatinib +

EGFR(del19), IC50: 39.9 nM

EGFR(C797S/T790M/del19), IC50: 67.2 nM

ALK,FLT3 {[allProObj[0].p_purity_real_show]}
Avitinib ++++

EGFR L858R/T790M, IC50: 0.18 nM

BTK {[allProObj[0].p_purity_real_show]}
EAI045 {[allProObj[0].p_purity_real_show]}
Almonertinib {[allProObj[0].p_purity_real_show]}
BI-4020 ++++

EGFRdel19 T790M C797S, IC50: 0.2 nM

{[allProObj[0].p_purity_real_show]}
EGFR-IN-7 ++++

EGFRd746-750/T790M/C797S, IC50: 0.26 nM

EGFRL858R/T790M, IC50: 0.19 nM

{[allProObj[0].p_purity_real_show]}
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。

AG-825 实验方案

计算器
存储液制备 1mg 5mg 10mg

1 mM

5 mM

10 mM

2.52mL

0.50mL

0.25mL

12.58mL

2.52mL

1.26mL

25.16mL

5.03mL

2.52mL

AG-825 技术信息

CAS号149092-50-2
分子式C19H15N3O3S2
分子量 397.471
别名 Tyrphostin AG-825
运输蓝冰
存储条件

粉末 Sealed in dry,Store in freezer, under -20°C

液体 -20°C:3-6个月-80°C:12个月

溶解度

DMSO: 250 mg/mL(628.98 mM),配合低频超声助溶,注意:DMSO长时间开封后,会吸水并导致溶解能力下降,请避免使用长期开封的DMSO

动物实验配方
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