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货号 产品名 纯度
A1942326 现货 Zelasudil

Zelasudil是一种针对Rho相关蛋白激酶(ROCK)的有效抑制剂,具有ROCK2结合的高度亲和力,显示出在相关疾病研究中的应用潜力。

98%
A168750 现货 BAY-549

ROCK inhibitor is a highly potent inhibitor of human ROCK-1 and ROCK-2 isoenzymes with IC50 values of 0.6 and 1.1 nM, respectively.

99%+
A130094 现货 Ripasudil

K-115 HCl is potent ROCK inhibitor with IC50 of 51 nM and 19 nM for ROCK1 and ROCK2, respectively, used for the treatment of glaucoma and ocular hypertension.

99%+
A919821 现货 ROCK2-IN-2

ROCK2-IN-2 is a selective ROCK2 inhibitor extracted from patent US20180093978A1, Compound A-30, has an IC50 of <1 μM.

99%+
A317869 现货 RKI-1447

RKI-1447 is a potent small molecule inhibitor of ROCK1 and ROCK2, with IC50 of 14.5 nM and 6.2 nM, respectively, and has anti-invasive and antitumor activities.

99%+
A1177078 现货 ROCK inhibitor-2

ROCK inhibitor-2是一种选择性 ROCK1ROCK2 双重抑制剂,IC50 分别为 17 nM 和 2 nM。该化合物可用于细胞骨架重塑、肿瘤转移及心血管疾病等研究领域,特别在细胞迁移和增殖的调控中具有应用潜力。

99%+
A1598869 现货 ROCK1-IN-1

ROCK1-IN-1是一种 ROCK1 抑制剂,用于高血压、青光眼和勃起功能障碍等相关研究。

95%
A1806913 现货 CAY10746

CAY10746是一种选择性 Rho 激酶 (ROCK) 抑制剂,对 ROCK I 和 ROCK II 的 IC50 分别为 0.014 μM 和 0.003 μM,广泛应用于糖尿病视网膜病变(DR)等与 ROCK 信号通路相关的疾病研究。

98%
A1229459 现货 ROCK-IN-5

ROCK-IN-5是一种有效的 ROCKERK、GSK 和 AGC 蛋白激酶的抑制剂,具有在增殖性、心脏和神经退行性疾病研究中的潜力。

99%+
A255643 现货 Belumosudil

Belumosudil (KD025) 是一种选择性 ROCK2 抑制剂,对 ROCK2IC50 值为 105 nM,对 ROCK1IC50 值为 24 µM,具有抗纤维化特性。

99%+
A105790 现货 GSK269962A HCl

GSK269962 HCl is a selective ROCK (Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.

99%+
A747327 现货 H-1152 2HCl/H-1152二盐酸盐

H-1152 2HCl, an isoquinolinesulfonamide derivative, is a more specific, stronger and membrane-permeable inhibitor of Rho-kinase with a Ki value of 1.6 nM, but poor inhibitor of other serine/threonine kinases.

99%
A112358 现货 Y-27632

Y-27632 是一种口服有效的、ATP 竞争性的 ROCK-I 和 ROCK-II 抑制剂,Ki 值分别为 220 nM 和 300 nM。

99%+
A204681 现货 Y-33075 2HCl/Y-39983盐酸

Y-33075 2HCl具有选择性作为 ROCK 抑制剂,IC50 为 3.6 nM。

99%+
A225129 现货 Narciclasine/水仙环素

Narciclasine is a plant growth modulator. Narciclasine modulates the Rho/Rho kinase/LIM kinase/cofilin signaling pathway, greatly increasing GTPase RhoA activity as well as inducing actin stress fiber formation in a RhoA-dependent manner.

99%+
A1263609 现货 Netarsudil Mesylate

Netarsudil Mesylate是一种 ROCK 激酶和去甲肾上腺素转运体的双重抑制剂,适用于眼科疾病的研究,尤其是在降低眼内压及治疗青光眼方面具有显著的作用。

99%+
A244270 现货 Hydroxyfasudil/羟基法舒地尔

Hydroxyfasudil, metabolite of Fasudil, is a potent Rho-kinase inhibitor and vasodilator.

99%+
A405951 现货 SR-3677

SR-3677 is a potent and selective ROCK-II inhibitor with an IC50 of ~3 nM in enzyme and cell based assays, and its IC50 for ROCK-I is 56 ± 12 nM.

99%
A552197 现货 Netarsudil hydrochloride

Netarsudil primarily targets cells in the conventional outflow tract, efficiently decreasing IOP in both human and non-human primate eyes.

99%+
A1549873 现货 RKI-1447 2HCl

RKI-1447 2HCl是一种有效的选择性 ROCK 抑制剂,对 ROCK1ROCK2IC50 分别为 14.5 和 6.2 nM。它能抑制结直肠癌细胞的生长并促进细胞凋亡

98%+
产品名 ROCK ROCK1 ROCK2 其他靶点 纯度
Thiazovivin +

ROCK, IC50: ~0.5 μM

98%
Netarsudil hydrochloride ++++

ROCK, Ki: 2 nM

99%+
Y-33075 2HCl ++++

ROCK, IC50: 3.6 nM

99%+
ROCK1-IN-1 ++

ROCK, Ki: 17nM

95%
GSK429286A +++

ROCK1, IC50: 14 nM

++

ROCK2, IC50: 63 nM

99%+
Ripasudil ++

ROCK1, IC50: 51 nM

++

ROCK2, IC50: 19 nM

99%+
Belumosudil ++

ROCK2, IC50: 60 nM

ROCK2, Ki: 41 nM

99%+
Y-27632 dihydrochloride ++

ROCK1, Ki: 140 nM

+

ROCK2, Ki: 300 nM

99%+
Fasudil HCl +

ROCK2, Ki: 330 nM

PKG,Rho 98%
Chroman 1 ++++

ROCK1, IC50: 52 pM

++++

ROCK2, IC50: 1 pM

99%
BAY-549 ++++

ROCK1, IC50: 0.6 nM

++++

ROCK2, IC50: 1.1 nM

99%+
AT13148 +++

ROCK1, IC50: 6 nM

+++

ROCK2, IC50: 4 nM

PKA 98+%
RKI-1447 +++

ROCK1, IC50: 14.5 nM

+++

ROCK2, IC50: 6.2 nM

99%+
Hydroxyfasudil HCl +

ROCK1, IC50: 0.73 μM

+

ROCK2, IC50: 0.72 μM

PKA 98%
H-1152 2HCl +++

ROCK2, IC50: 0.0120 μM

PKG 99%
GSK269962A HCl ++++

ROCK1, IC50: 1.6 nM

+++

ROCK2, IC50: 4 nM

99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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