AGN 192870是一种 RAR 中性拮抗剂，对 RARα、RARβ 和 RARγ 的 Kd 分别为 147 nM、33 nM 和 42 nM。它对 RARα 和 RARγ 的 IC50 分别为 87 nM 和 32 nM，并且对 RARβ 显示部分激动作用。

Liarozole (R75251; R85246)是一种咪唑衍生物，作为口服有效的维甲酸 (RA) 代谢阻断剂 (RAMBA)，它抑制维甲酸依赖的细胞色素P450 (CYP26) 4-羟基化，IC50为7 μM，从而增加组织维甲酸水平，并具有抗肿瘤特性。

HX 531 is a potent RXR antagonist with IC50 of 18 nM.

(R)-Flurbiprofen is the R-enantiomer of the racemate NSAID flurbiprofen, inhibiting the binding of [3H]9-cis-RA to RXRαLBD with IC50 of 75 μM.

4-Hydroxyretinoic acid是一种天然的类视黄酸衍生物，通过结合核受体 RAR 和 RXR-alpha，调控基因表达、促进细胞分化，并诱导癌细胞凋亡，同时具有免疫调节和神经保护等多种生理作用。

SR11237 (BMS-649)是一种选择性的视黄酸 X 受体 (RXR) 激动剂，无视黄酸受体 (RAR) 活性。它诱导 RXR/RXR 同源二聚体的形成，并激活含 RXR 响应元件的报告基因。

Acitretin is an analog of retinoid that can activate α-secretase ADAM10 gene expression. It has been used in the treatment of severe psoriasis.

DM1-SMe 是 IMGN901 中 Maytansinoid 的非结合形式。在一组人类肿瘤细胞系中，DM1-SMe 比母体 Maytansinoid 强效约 3-10 倍，IC50 值在 0.003 到 0.01 nM 之间

Trifarotene is a retinoic acid receptor (RAR) agonist with Kdapp of 2, 15 and 500 nM for RARγ, RARβ and RARα, respectively.

CH-55 is a potent agonist for RAR-α and RAR-β receptors.

Palovarotene is a selective retinoic acid receptor gamma (RAR-γ) agonist for the treatment of emphysema.

Amsilarotene (TAC-101; Am 555S) 是一种口服活性的合成类视黄醇，对视黄酸受体 α (RAR-α) 具有选择性亲和力，诱导多种癌细胞凋亡，可用于癌症研究。

UVI 3003 is a potent and selective RXR antagonist, used as a tool to test the contribution of RXR to transactivation by a given RXR heterodimer.

All trans-Retinal, a component of the retinoid cycle, is converted to retinoic acid in vivo by the action of retinal dehydrogenase. Retinoic acid is a ligand for both RAR and RXR. All trans-retinal ias a potent photosensitizer.

AGN 193109 is a high affinity pan-retinoic acid receptor (RAR) antagonist with Kds of 2, 2 and 3 nM at RARα, RARβ and RARγ, respectively.

Magnolol is a multifunctional compound isolated from the Chinese medicinal plant Magnolia officinalis, with antifungal, antibacterial and antioxidant effects, as well as anti-inflammatory activity by interferring with NF-κB signaling and inhibiting IL-6-induced STAT3 activation.

AC55649 is an agonist of the retinoic acid receptor β (RAR-β).

AR7 is a retinoic acid receptor α (RARα) antagonist.

LG-100064 is an agonist of RXRα, RXRβ and RXRγ with EC50s of 330 nM, 200 nM, and 260 nM, respectively.

Tazarotene selectively binds to retinoic acid receptors RAR-β and RAR-γ, it is the first receptor-selective aromatic retinoid that has effective treatment for psoriasis, hemorrhoids.