Glycopyrrolate is a muscarinic competitive antagonist used as an antispasmodic.

Captopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM.

Benazepril HCl is an ACE inhibitor, primarily used in treatment of hypertension. Benazepril HCl is the HCl form of Benazepril.

Irbesartan is a selective and competitive nonpeptide angiotensin II antagonist with antihypertensive activity.

Cilnidipine is a dual L- and N-type calcium channel blocker with antihypertensive, sympatholytic and neuroprotective activity.

Diltiazem HCl is a benzothiazepine derivative with vasodilating action due to its antagonism of the actions of the calcium ion in membrane functions.

Flavoxate HCl is a competitive AChR antagonist with IC50 of 12.2 μM, used as a muscle relaxant.

Fluvoxamine maleate is a selective serotonin reuptake inhibitor and can be used as an antidepressant.

Nitrendipine is a dihydropyridine calcium channel blocker with an IC50 of 95 nM.

Terazosin HCl is a selective antagonist for alpha-adrenergic receptor, used for treatment for hypertension and prostate enlargement (BPH) through lowering the blood pressure with elimination half-life of ‎12 hours.

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker.

Etodolac is a non-selective inhibitor of COX with IC50 of 53.5 nM, it is a non-steroidal anti-inflammatory compound.

Phentolamine mesylate is a reversible and nonselective alpha-adrenergic receptor antagonist, used for the prevention or control of hypertensive episodes.

Doxazosin mesylate is a selective α1-adrenergic receptor blocker, used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH).

Flutamide is a competitive non-steroidal antagonist of androgen receptor.

Minoxidil is an antihypertensive vasodilator medication.

Valsartan is a selective angiotensin II AT1 receptor antagonist with elimination half-life‎ of ‎6 hours.

Nifedipine 是一种钙通道阻滞剂，对 L-型钙通道具有高亲和力，IC50 值为 10 nM。Nifedipine 具有抗高血压和抗心绞痛作用，可用于心血管疾病的研究。

Reserpine is a naturally occuring brain-penetrant and irreversible VMAT (vesicular monoamine transporter 1 and 2) antagonist.

Famotidine is antagonist of histamine H2–receptor with IC50 of 0.6 mM that used to treat heartburn and other digestive conditions.