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货号 产品名 纯度
A602643 现货 E 64c

Loxistatin acid, a derivative of E-64, is an irreversible and membrane-permeant cysteine protease inhibitor.

95%
A1147307 现货 Cruzain-IN-1

Cruzain-IN-1是一种针对克鲁斯氏锥体虫半胱氨酸蛋白酶 (Cruzain)的抑制剂,通过共价结合实现高效抑制,为寄生虫病治疗提供了新的途径。

99%+
A120064 现货 NSC 185058

NSC 185058 is an ATG4B inhibitor with IC50 of 3.24 µM.

99%+
A590110 现货 Calpeptin/钙肽素

Calpeptin is a potent, cell-permeable calpain inhibitor with ID50 of 52 nM, 34 nM, 138 nM, and 40 nM for Calpain I (porcine erythrocytes), Calpain II (porcine kidney), Papainb, and Calpain I (human platelets), respectively.

98%+
A175883 现货 N-Ethylmaleimide/N-乙基马来酰亚胺

N-Ethylmaleimide is an irreversible inhibitor of all cysteine peptidases, it's an organic compound derived from maleic acid.

97%
A663950 现货 Leupeptin hemisulfate/亮抑酶肽半硫酸盐

Leupeptin Hemisulfate is a reversible serine/cysteine protease inhibitor, inhibits cathepsins B, H, L, and S, calpain, and trypsin.

97%
A473978 现货 LY 3000328

LY 3000328 is a highly selective and potent Cathepsin S inhibitor with IC50 of 7.7±5.85 nM and 1.67±1.17 nM for hCat S and mCat S respectively, can be used in treatment for abdominal aortic aneurysm.

99%+
A544458 现货 TPCK

TPCK is a non-specific irreversible inhibitor of serine/cysteine proteases. It acts by inhibiting ScRce1 in the presence of a Ras reporter, but not in the presence of the a-factor peptide.

98%
A254787 现货 Balicatib/巴利卡替

Balicatib is a potent and selective inhibitor of cathepsin K ,with 10-100 fold more potent in cell-based enzyme occupancy assays than against cathepsin B, L, and S.

98%+
A328069 现货 Odanacatib/奥当卡替

Odanacatib is a potent, selective, and neutral inhibitor of cathepsin K (human/rabbit) with IC50 of 0.2 nM/1 nM, and demonstrated high selectivity versus off-target cathepsin B, L, S.

99%+
A917874 现货 CA-074 methyl ester

CA-074 methyl ester是一种特异性的半胱氨酸蛋白酶B抑制剂,具有神经保护、抗癌和抗炎等强效生物活性。

95%
A158847 现货 MG-101/钙蛋白酶抑制剂I

MG-101 is a potent inhibitor of cysteine proteases including calpain I (Ki = 190 nM), calpain II (Ki = 220 nM), cathepsin B (Ki = 150 nM), and cathepsin L (Ki = 500 pM).

98%+
A252147 现货 E-64/蛋白酶抑制剂E 64

E-64(蛋白酶抑制剂E 64)是一种高效的不可逆广谱半胱氨酸蛋白酶抑制剂,对木瓜蛋白酶的IC50为9 nM。

99%+
A162425 现货 E-64d/阿洛司他丁

E-64d(E64d)是一种细胞可渗透、不可逆的广谱半胱氨酸蛋白酶抑制剂,对MERS-CoV具有入侵阻断作用。

99%+
A793997 现货 Cysteine Protease inhibitor hydrochloride

Cysteine protease inhibitor HCl is an inhibitor of cysteine protease.

99%+
A767839 现货 PMSF/苄基磺酰氟

PMSF is a non-selective serine/cysteine protease inhibitor, also blocks anandamide metabolism.

95%
A257707 Aureusimine B

98+%
A686967 PD150606

PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively).

98%
A812592 Cysteine Protease inhibitor/半胱氨酸蛋白酶抑制剂

Cysteine protease inhibitor is an inhibitor of cysteine protease.

99%
A2794868 E 64c

99%
产品名 Cysteine Protease 其他靶点 纯度
Z-FA-FMK 99%+
Leupeptin hemisulfate 97%
PMSF 95%
PD 151746 +

μ-Calpain, IC50: 260 nM

m-calpain, IC50: 5.33 μM

98%
Odanacatib ++++

Cathepsin K (human), IC50: 0.2 nM

Cathepsin K (rabbit), IC50: 1 nM

99%+
E-64 +++

Cysteine protease, IC50: 9 nM

99%+
E 64c 95%
E-64d 99%+
MG-101 98%+
Calpeptin ++

Calpain I (porcine erythrocytes), ID50: 52 nM

Calpain II (porcine kidney), ID50: 40 nM

98%+
Cathepsin inhibitor 1 +++

Cathepsin L2, pIC50: 5.5

Cathepsin L, pIC50: 7.9

98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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