Fluvastatin Sodium is a synthetic indole-heptanoic-acid-derived inhibitor of hepatic HMG-CoA reductase with IC50 of 8 nM.

Enalaprilat is the first dicarboxylate-containing ACE inhibitor with IC50 of 1.94 nM, which is the active metabolite of enalapril.

Perindopril erbumine Perindopril is a long-acting ACE inhibitor with IC50 of 1.05 nM, used in treatment for hypertension.

Captopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM.

Benazepril HCl is an ACE inhibitor, primarily used in treatment of hypertension. Benazepril HCl is the HCl form of Benazepril.

Bezafibrate is the agonist of PPAR and the EC50 for PPAR⍺, PPARβ, PPARẟ is 50 , 20, and 60 nM respectively. It has hypolipidemic effect.

Lisinopril is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks.

Clofibrate, a fibric acid derivative, is a selective agonist of peroxisome proliferator-activated receptor α (PPARα) with EC50 of 50 µM. Clofibrate has been used to treat hyperlipoproteinemia type III and severe hypertriglyceridemia.

Rosuvastatin Calcium is a competitive and synthetic HMG-CoA reductase inhibitor with IC50 value of 11 nM.

Candesartan Cilexetil is a benzimidazole-derived and competitive AT1 inhibitor with IC50 value of 0.26 nM.

Amlodipine Besylate is a long-acting calcium channel blocker used to lower blood pressure and prevent chest pain.

Gemfibrozil is an agonist of PPARα. It can act as a hyperlipidemic agent that elevates plasma HDL and lowers triglycerides.

Mevastatin is the first discovered statin-class HMG-CoA reductase inhibitor used as a cholesterol-lowering agent isolated from Penicillium citinium.

Telmisartan是一种高效且长效的血管紧张素II 1型受体（AT1）拮抗剂，选择性抑制125I-AngII与AT1受体结合，IC50为9.2 nM。

Ciprofibrate is an agonist of peroxisome proliferator-activated receptor PPAR⍺. It is used in dyslipidaemia.

Lovastatin是一种用于降低胆固醇的细胞渗透性 HMG-CoA 还原酶抑制剂。

Manidipine 2HCl is a L/T-type calcium channel blocker for Ca2+ current with IC50 of 2.6 nM.

Probucol is a synthetic antioxidant used to lower the level of cholesterol in the bloodstream by increasing the rate of LDL catabolism.

Ramiprilat,the active metabolite of Ramipril, is a non-sulfhydryl angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.

Atorvastatin hemicalcium salt（CI-981）是一种口服活性的3-羟基-3-甲基戊二酰辅酶A（HMG-CoA）还原酶抑制剂，有效降低血脂。它抑制人SV-SMC增殖和侵袭的IC50值分别为0.39 μM和2.39 μM。