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Oxytocin是一种多效性神经垂体激素,参与分娩、哺乳和亲社会行为的调节。它具有抗炎、抗氧化和保护作用,尤其在面对创伤或逆境时。Oxytocin 可用作研究压力应对和神经生物学的模型分子。
LIT-001是首个非肽类催产素受体 (OT-R) 激动剂,EC50为55 nM,Ki值为226 nM。
Cligosiban是一种口服有效的高选择性催产素受体拮抗剂,Ki为9.5 nM,用于抑制啮齿动物的生理性射精,具有良好的药代动力学特性。
Oxytocin acetate是一种哺乳动物神经垂体激素,通过特异性的、高亲和力的催产素受体介导其作用,是催产素受体的配体。
Atosiban acetate是一种宫缩抑制剂,可通过抑制催产素介导的肌层细胞钙离子释放,达到快速抑制子宫收缩的效果,常用于治疗早产。
Atosiban是一种九肽类加压素/催产素受体拮抗剂,可用作宫缩抑制剂,用于自发性早产的研究和治疗。
Lysipressin is an antidiuretic hormone that havs been found in pigs and some marsupial families. It can induce contraction of the rabbit urinary bladder smooth muscle.
L-368,899 HCl is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively, used as a tocolytic agent.
OT-R antagonist 1 is a potent and selective nonpeptide low molecular weight OT-R antagonist.
SHR1653 is a highly potent oxytocin receptor antagonist with excellent blood-brain barrier penetration. It might be beneficial for the treatment of CNS-related premature ejaculation.
OT antagonist 1 (Compound 4) is a potent, selective Oxytocin antagonist with a Ki of 50 nM.
Retosiban is an oral active, potent and selective, sub-nanomolar (Ki = 0.65 nM) oxytocin receptor antagonist with > 1400-fold selectivity over the related vasopressin receptors. Retosiban inhibits the procontractile effect of stretch on human myometrium and prevent stretch-induced stimulation of human myometrial contractility.
GSK 557296 is a potent, selective and orally bioavailable oxytocin receptor antagonist, with a pKi of 9.9 for human oxytocin receptor.
OT-R antagonist 2 is a nonpeptide low molecular weight OT-R antagonist.
OT antagonist 3 is an oxytocin (OT) antagonist extracted from patent WO2007017752A1.
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth and an agonist at peripheral oxytocin receptors.
Tags: OXTR | G蛋白偶联受体/G蛋白 | GPCR/G Protein | OXTR 相关产品
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