Pirodavir is the prototype of a class of broad-spectrum antipicornavirus compounds and a potent human rhinovirus (HRV) capsid-binding inhibitor.

Tilorone 2HCl is an orally active interferon inducer, used as an antiviral drug.

1-[(2R,3S,4R,5R)-3-Fluoro-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-5-iodopyrimidine-2,4-dione是一种具有抗病毒活性的核苷类似物。Fialuridine 具有抗正痘病毒活性。

2′,3′-Dideoxyadenosine is a nucleoside analog of deoxyadenosine. It inhibits adenylyl cyclase and may play a key role in the inhibition of tumor progression. It is a potent inhibitor of reverse transcriptase enzyme of HIV.

Atazanavir Sulfate is a protease inhibitor used as an antiretroviral medication to treat and prevent HIV/AIDS.

Trifluorothymidine is a derivative of thymidine that can inhibit thymidylate synthase and lead to DNA damage and apoptosis. It could be used to treat colorectal cancer.

Mizoribine is an immunosuppressive agents (IC50=100 μM) that inhibit the proliferation of lymphocytes selectively, via inhibition of IMPDH.

Etravirine is an inhibitor of non-nucleoside reverse transcriptase used to treat HIV.

Peramivir Trihydrate is a novel cyclopentane neuraminidase inhibitor of influenza virus, used to treat acute symptomatic influenza A and B.

Valacyclovir HCl is a Herpes Simplex Virus and Herpes Zoster Virus nucleoside analog DNA polymerase inhibitor as it is a synthetic purine nucleoside analogue.

Plerixafor is a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM, respectively.

Efavirenz is an inhibitor of wild-type HIV-1 reverse transcriptase with Ki of 2.93 nM and the IC95 of its replicative spread is 1.5 nM in cell culture.

Oseltamivir（GS 4104）是一种口服活性的流感病毒神经氨酸酶抑制剂（NAI）。它有效抑制流感A/H3N2、A/H1N2、A/H1N1和B病毒，平均IC50值分别为0.67 nM、0.9 nM、1.34 nM和13 nM。

Sofosbuvir（GS-7977）是一种HCV RNA复制抑制剂，EC50为92 nM。

α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity.

Entecavir, an analogue of guanosine, is reverse transcription inhibitor of HBV with EC50 of 3.75 nM in HepG2 cell.

Lopinavir（ABT-378）是一种高效选择性的HIV-1蛋白酶抑制剂，对野生型和突变型HIV蛋白酶的Ki值在1.3至3.6 pM之间。其作用是阻止HIV-1的成熟，从而阻止其感染性。Lopinavir还表现出对SARS-CoV 3CLpro的抑制作用，IC50为14.2 μM。

Decitabine is a potent inhibitor of DNA methyltransferase with IC50 of 438 nM and 4.38 nM in HL-60 and KG1a cells, respectively.

Lamivudine is a potent nRTI (nucleoside analog reverse transcriptase inhibitor) an analogue of cytidine,which can inhibit both HIV 1 and 2 reverse transcriptase as well as the reverse transcriptase of hepatitis B.

Vidarabine is an antiviral drug effects by interfering with the synthesis of viral DNA, which is used in treatment of herpes simplex and varicella zoster viruses.