Eprobemide is a reversible monoamine oxidase A inhibitor and is classified as a drug for depression.

Harmane是一种β-咔啉生物碱，具有显著的神经毒性及MAO A/B抑制活性，适用于研究神经毒性、MAO抑制和相关生物学过程。

BU224 HCl是一种高选择性、高亲和力的咪唑啉 I2 受体配体 (Ki = 2.1 nM)，常作为 I2 受体拮抗剂，具有神经保护、抗炎和抗凋亡作用，可用于阿尔茨海默病等神经退行性疾病的研究。

BU226 HCl是一种高效、选择性咪唑啉 2 (I2) 受体配体，对I2受体的结合力强 (Ki = 1.4 nM)，而对I1受体的亲和力显著较低 (IC₅₀ = 534.5 nM)。该化合物在抗抑郁机制研究中展现了潜在的应用价值。

Rilmenidine Phosphate is an oxazole-derived agonist of adrenergic receptor α2 and Imidazoline receptor, used in trials studying the treatment of hypertension and chronic kidney disease.

Moxonidine is a selective agonist of imidazoline I1 receptors and alpha-2 receptor used as an antihypertensive drug.

Moxonidine HCl is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.

Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively.