(R)-Equol is an agonist of both ERα and ERβ with Kis of 27.4 and 15.4 nM, respectively.

Lasofoxifene is a non-steroidal selective estrogen receptor modulator (SERM).

Estradiol cypionate is a synthetic ester. Compared to other commonly used estradiol esters, via the intramuscular route, estradiol cypionate is found to have the longest duration of action with a duration of ~11 days,

PCO371 is an orally active full agonist of parathyroid hormone receptor 1 (PTHR1), shows no effect on PTH type 2 receptor.

Segetalin B是从Vaccaria segetalis中分离得到的一种环五肽，具有类雌激素活性。

NH-3是一种具有口服活性的、可逆的甲状腺激素受体 (THR) 拮抗剂，IC50 值为 55 nM。它是选择性甲状腺素 GC-1 的衍生物，能够阻止甲状腺激素与其受体的结合，并抑制辅因子的招募。

FLTX1是一种荧光他莫昔芬 (Tamoxifen) 衍生物，可在透化和非透化条件下特异性标记细胞内他莫昔芬结合位点 (雌激素受体)。FLTX1 在乳腺癌细胞中显示出他莫昔芬有效的抗雌激素特性，且不对子宫产生雌激素激动作用。

Palazestrant是一种抗雌激素药物，具有抗肿瘤作用，常与 HER2 抑制剂联合使用，以抑制 ER+/HER2+ 类型的癌症。

SLU-PP-332是一种泛雌激素受体相关受体 (ERR) 激动剂，可增强线粒体功能及细胞呼吸，广泛用于代谢性疾病及肌肉功能改善的研究。

β-Estradiol 17-Heptanoate 是一种短效雌激素，与 dihydroxyprogesterone acetophenide 组合，可用作每月注射的避孕药。

Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM), with a pIC50 of 0.46. It has been found to be both estrogenic and antiproliferative in ER-positive endocrine-resistant breast cancer cell lines that overexpress protein kinase C alpha (PKCα).

4,4'-Iminodiphenol 是一种基于二苯胺骨架的无活性雌激素受体配体。

Elacestrant 2HCl is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities.

AC 186 is a potent and selective ERβ agonist with EC50 of 6 nM.

LCS3是一种谷胱甘肽二硫化物还原酶 (GSR) 和硫氧还蛋白还原酶1 (TXNRD1)抑制剂，表现出抗肿瘤活性，并可用于诱导肺腺癌细胞凋亡。

AZD-9833 is a potent and orally active estrogen receptor (ER) antagonist. AZD-9833 is used for the study of ER+ HER2-advanced breast cancer[1].

XCT-790 is an agonist of estrogen related receptor alpha (ERRα) and can induce death of cancer cells resistant to chemotherapy.

PHTPP has selective antagonism of estrogen ERβ receptor .

Endoxifen E-isomer HCl is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).

Eprotirome is a liver-selective thyroid hormone receptor agonist.