Asenapine Maleate is a 5-HT and dopamine D2 receptor antagonist used to treat schizophrenia and bipolar mania.

BMY 7378 2HCl is a 5-HT1A partial agonist and a high-affinity α1D adrenoceptor antagonist with Ki values of 2, 800 and 600 nM for cloned rat α1D, rat α1A and hamster α1B receptors respectively.

Naftopidil is a selective α1-adrenergic receptor antagonist or α blocker used for treatment for lower urinary tract symptoms (LUTS) due to benign prostatic hyperplasia (BPH).

Naftopidil 2HCl is a selective α1-adrenergic receptor antagonist or α blocker used for treatment for lower urinary tract symptoms (LUTS) due to benign prostatic hyperplasia (BPH).

Doxazosin mesylate is a selective α1-adrenergic receptor blocker, used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH).

Alfuzosin HCl is an antagonist of α1 adrenergic receptor used to treat benign prostatic hyperplasia (BPH).

Silodosinis a selective prostate α1-adrenoceptor antagonist for symptomatic treatment of benign prostatic hyperplasia.

Phentolamine mesylate is a reversible and nonselective alpha-adrenergic receptor antagonist, used for the prevention or control of hypertensive episodes.

Prazosin HCl is a selective α-1-adrenergic receptor antagonist used to treat hypertension, anxiety, and posttraumatic stress disorder (PTSD).

Terazosin HCl is a selective antagonist for alpha-adrenergic receptor, used for treatment for hypertension and prostate enlargement (BPH) through lowering the blood pressure with elimination half-life of ‎12 hours.

Phenoxybenzamine HCl is a non-selective irreversible dibenzamine α adrenergic antagonist with antihypertensive and vasodilatory properties.

Atipamezole is a synthetic competitive α2 adrenergic receptor antagonist with Ki value of 1.6 nM.

Tolazoline HCl is a competitive non-selective α-adrenergic receptor antagonist, used as a a vasodilator directly acting on blood vessels and also increasing cardiac output.

Yohimbine HCl is naturall occuring alpha-2 adrenergic antagonist derived from the bark of the African tree Pausinystalia johimbe, used as a veterinary drug to reverse sedation in dogs and deer.

Piribedil is an antiparkinsonian agent and piperazine derivative which acts as a D2 and D3 receptor agonist.