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Theophylline-7-acetic Acid
茶碱乙酸 /Theophylline-7-acetic Acid
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货号：A229005
同义名：
Acefylline;Theophyllineacetic acid
Theophylline-7-acetic Acid 是一种腺苷受体拮抗剂，具支气管扩张和心脏刺激作用，可用于哮喘的研究。
Theophylline-7-acetic Acid 化学结构
Theophylline-7-acetic Acid 3D分子结构
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Theophylline-7-acetic Acid 纯度/质量文件 产品仅供科研
货号：A229005
标准纯度：
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Theophylline-7-acetic Acid 质控信息
ZM241385
✔
99%+
Istradefylline
+++
Adenosine A2A receptor, Ki: 2.2 nM
98%
Reversine
+
human A3 adenosine receptor, Ki: 0.66 μM
98%
SCH58261
++++
bovine A2a, Ki: 2.0 nM
rat A2a, Ki: 2.3 nM
99%+
A2A receptor antagonist 1
++
A1R, Ki: 264 nM
A2AR, Ki: 4 nM
99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
Theophylline-7-acetic Acid 生物活性
描述
Acefylline (Theophyllineacetic acid), a xanthine derivative, is an adenosine receptor antagonist. Theophylline (THEO) and its xanthinic derivatives inhibit lung phosphodiesterase (PDE) and block adenosine receptors in the induction of bronchodilatation[3] [4]
Theophylline-7-acetic Acid 参考文献
[1] Mechin MC, Cau L, et al. Acefylline activates filaggrin deimination by peptidylarginine deiminases in the upper epidermis. J Dermatol Sci. 2016 Feb;81(2):101-6.
[2] Voynikov Y, Valcheva V, et al. Theophylline-7-acetic acid derivatives with amino acids as anti-tuberculosis agents. Bioorg Med Chem Lett. 2014 Jul 15;24(14):3043-5.
[3] Ferretti C, Coppi G, Blengio M, Genazzani E. Inhibitory effect of theophylline, theophylline-7-acetic acid, ambroxol and ambroxol-theophylline-7-acetate on rat lung cAMP phosphodiesterase isoenzymes. Int J Tissue React. 1992;14(1):31-6
[4] Méchin MC, Cau L, Galliano MF, Daunes-Marion S, Poigny S, Vidaluc JL, Bessou-Touya S, Takahara H, Serre G, Duplan H, Simon M. Acefylline activates filaggrin deimination by peptidylarginine deiminases in the upper epidermis. J Dermatol Sci. 2016 Feb;81(2):101-6
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Theophylline-7-acetic Acid 实验方案
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1mg
5mg
10mg
1 mM
5 mM
10 mM
4.20mL
0.84mL
0.42mL
20.99mL
4.20mL
2.10mL
41.98mL
8.40mL
4.20mL
Theophylline-7-acetic Acid 技术信息
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