JNJ-1661010 is a selective inhibitor of FAAH with IC50 of 10 nM (rat) and 12 nM (human).

MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.

CB2R/FAAH modulator-2是一种双重靶向调节剂，既作为 CB2R 激动剂 (Ki = 10.8 nM) 又作为 FAAH 抑制剂 (IC₅₀ = 6.2 μM)。该化合物适用于癌症、神经退行性疾病中的有害炎症反应调控以及 COVID-19 感染相关的炎症研究。

AA38-3是一种丝氨酸水解酶 (SH) 抑制剂，能够有效抑制ABHD6、ABHD11和FAAH三种SHs。这使得它在脂质代谢和神经保护研究中具有应用前景。

N-(3-Methoxybenzyl)palmitamide, found in lepidium meyenii walp., is a promising inhibitor of fatty acid amide hydrolase (FAAH). It could counteract the toxicity produced by Aβ (25-35).

AM 374是一种脂肪酸酰胺水解酶 (FAAH) 抑制剂，IC₅₀ 为 13 nM。该化合物常用于神经系统疾病的研究，尤其是与脂肪酸信号通路相关的疾病研究中。

LY2183240 is a highly potent blocker of anandamide uptake (IC50 = 270 pM).

URB937 is a FAAH inhibitor and increases anandamide levels, with an IC50 of 26.8 nM. URB937 fails to affect FAAH activity in the brain .

FAAH inhibitor 1 is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18±8 nM.

Macamide B is a natural product isolated and purified from the herbs of Lepidium meyenii Walp.

PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.

PF-04457845 selectively inhibits FAAH with an IC50 of 7.2 nM. It has anti-inflammatory effects and is used as analgesic.

URB-597 is fatty acid amide hydrolase (FAAH, IC50 = 4.6 nM) inhibitor without effect on other cannabinoid-related targets.

PF-750 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor with IC50 of 16.2 nM.

JZL195 functions as a dual inhibitor of FAAH and MAGL with IC50 of 13 nM and 19 nM respectively in brain of mouse.

CB2R/FAAH modulator-3是一种双重靶向调节剂，作为 CB2R 激动剂和 FAAH 抑制剂，作用于 CB2R 和 CB1R 的 Ki 值分别为 20.1 和 67.6 nM，对 FAAH 的 IC50 值为 3.4 μM，可用于癌症、神经退行性疾病中的有害炎症级联反应以及 COVID-19 感染相关研究。

VU534是一种NAPE-PLD激动剂，其EC50为0.30 μM。它是FAAH和sEH的双重抑制剂（IC50值为1.2 μM）。VU534通过NAPE-PLD依赖性途径增强巨噬细胞的吞噬作用，并在心血管代谢性疾病的研究中具有潜力。

MAGL-IN-5是一种非选择性的脂肪酶抑制剂，能够抑制单酰基甘油脂肪酶 (MAGL)、激素敏感脂肪酶 (HSL) 和脂肪酸酰胺水解酶 (FAAH)，IC₅₀ 值分别为 144、90 和 14 nM，常用于脂质代谢和神经退行性疾病研究。

Biochanin A 是一种天然异黄酮，是脂肪酸酰胺水解酶 (FAAH) 抑制剂，具有抗氧化、抗炎和抗癌作用。Biochanin A 主要用于癌症预防和治疗的研究。

BIA10-2474 is an inhibitor of fatty acid amide hydrolase (FAAH) with IC50 of 4.9 nM.