LY294002 是一种 PI3K 抑制剂，抑制 PI3Kα, PI3Kδ 和 PI3Kβ 的 IC50 分别为 0.5, 0.57, 0.97 μM。LY294002 具有抗肿瘤作用，可用于研究 PI3K/AKT 信号通路和相关癌症治疗。

Silmitasertib 是一种选择性的 CK2 抑制剂，对 CK2 具有高亲和力，对 CK2α 和 CK2α' 的 IC50值均为 1 nM。Silmitasertib 具有抗肿瘤和抗炎作用，主要用于癌症和炎症相关疾病的研究。

DMAT is a potent and specific CK2 inhibitor with an IC50 value of 130 nM.

GO289 is a potent and selective CK2 inhibitor.

BioE-1115 is a highly selective and potent PAS kinase (PASK) inhibitor with an IC50 of ~4 nM. BioE-1115 is also a potent casein kinase 2α inhibitor with an IC50 of ~10 μM .

Silmitasertib sodium salt是一种口服可用的、高选择性和高效的CK2抑制剂，对CK2α和CK2α'的IC50值均为1 nM。

TTP 22 is a high affinity, ATP-competitive casein kinase 2 (CK2) inhibitor with IC50/Ki of 0.1 μM/40 nM, showing selectivity for CK2 over JNK3, ROCK1, and MET (IC50> 10 μM).

TBB is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2)with IC50s of 0.9 and 1.6 μM for rat liver and human recombinant CK2 respectively).

DRB is a chemical compound that inhibits transcription elongation by RNA Polymerase II. It works as a transcription inhibitor.