Pristimerin是一种高效的单甘油脂肪酶 (MGL) 可逆抑制剂，IC50 为 93 nM。

Triptonide, a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f. with antileukemic, antitumor, anti-inflammatory activities, is effective in the treatment of autoimmune diseases. Triptonide can effectively inhibit canonical Wnt/β-catenin signaling by targeting the downstream C-terminal transcription domain of β-catenin or a nuclear component associated with β-catenin.

Triptolide, a diterpene triepoxide extracted from the Chinese herb Tripterygium wilfordii, functions as a NF-κB inhibitor with dual actions by disruption of p65/CBP interaction and by reduction of p65 protein.

Wilforgine is a natural product isolated and purified from the roots of Tripterygium wilfordii Hook. f. showing insecticidal activity of some degree.

Triptophenolide is a colorless crystalline plate isolated from ethyl acetate extracts of Tripterygium wilfordii.

Demethylzeylasteral, a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f., has strong immunosuppressive activity, that can be used in the fields of organ transplantation and autoimmune disorders. It increases both activation and inactivation time constants of Ca(2+) currents, and inhibits significantly the sperm acrosome reaction initiated by progesterone.

Wilforine is a natural product isolated and purified from the vines of Tripterygium wilfordii, with insecticidal activity by inhibiting the Na+-K+-ATPase in the central nervous system, and anti-inflammatory effect, which might be mediated by down-regulation of the expression of inflammatory factors TNF-α,IL-6 and NO.

Wilforlide A is a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f. with obvious anti-inflammatory effect.

Tripterifordin, a natural product isolated and purified from the roots of Tripterygium wilfordii, shows anti-HIV replication activity in H9 lymphocyte cells with an EC50 of 1 mg/mL.

Triptobenzene H is a natural product isolated and purified from the roots of Tripterygium wilfordii Hook.f. showing significant immunosuppressive activity.