Pristimerin是一种高效的单甘油脂肪酶 (MGL) 可逆抑制剂，IC50 为 93 nM。

Triptonide, a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f. with antileukemic, antitumor, anti-inflammatory activities, is effective in the treatment of autoimmune diseases. Triptonide can effectively inhibit canonical Wnt/β-catenin signaling by targeting the downstream C-terminal transcription domain of β-catenin or a nuclear component associated with β-catenin.

Triptolide, a diterpene triepoxide extracted from the Chinese herb Tripterygium wilfordii, functions as a NF-κB inhibitor with dual actions by disruption of p65/CBP interaction and by reduction of p65 protein.

Wilforgine is a natural product isolated and purified from the roots of Tripterygium wilfordii Hook. f. showing insecticidal activity of some degree.

Triptophenolide is a colorless crystalline plate isolated from ethyl acetate extracts of Tripterygium wilfordii.

Wilforine is a natural product isolated and purified from the vines of Tripterygium wilfordii, with insecticidal activity by inhibiting the Na+-K+-ATPase in the central nervous system, and anti-inflammatory effect, which might be mediated by down-regulation of the expression of inflammatory factors TNF-α,IL-6 and NO.

Wilforlide A is a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f. with obvious anti-inflammatory effect.

Tripterifordin, a natural product isolated and purified from the roots of Tripterygium wilfordii, shows anti-HIV replication activity in H9 lymphocyte cells with an EC50 of 1 mg/mL.

Triptobenzene H is a natural product isolated and purified from the roots of Tripterygium wilfordii Hook.f. showing significant immunosuppressive activity.