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N-Desmethyl-Apalutamide
N-Desmethyl-Apalutamide
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货号：A1364782
N-Desmethyl-Apalutamide 是 Apalutamide 的活性代谢产物，作用力约为原药物的三分之一。它由 CYP2C8 和 CYP3A4 介导形成，具有中等至强的 CYP3A4 和 CYP2B6 诱导作用，且与血浆蛋白 结合能力较强，适用于雄激素 受体
There will be a HazMat fee per item when shipping a dangerous goods. The HazMat fee will be charged to your UPS/DHL/FedEx collect account or added to the invoice unless the package is shipped via Ground service. Ship by air in Excepted Quantity (each bottle), which is up to 1g/1mL for class 6.1 packing group I or II, and up to 25g/25ml for all other HazMat items.
Type HazMat fee for 500 gram (Estimated) Excepted Quantity USD 0.00 Limited Quantity USD 15-60 Inaccessible (Haz class 6.1), Domestic USD 80+ Inaccessible (Haz class 6.1), International USD 150+ Accessible (Haz class 3, 4, 5 or 8), Domestic USD 100+ Accessible (Haz class 3, 4, 5 or 8), International USD 200+
N-Desmethyl-Apalutamide 化学结构
N-Desmethyl-Apalutamide 3D分子结构
规格
价格
会员价
库存
数量
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N-Desmethyl-Apalutamide 纯度/质量文件 产品仅供科研
货号：A1364782
标准纯度：
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产品说明书
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N-Desmethyl-Apalutamide 质控信息
Cyproterone acetate
++++
Androgen Receptor, IC50: 7.1 nM
98%
Apalutamide
+++
Androgen Receptor, IC50: 16 nM
98%
AZD3514
+
Androgen Receptor, Ki: 2.2 μM
98%
Darolutamide
++++
Androgen receptor, Ki: 11 nM
98%
Flutamide
+++
Androgen Receptor, Ki: 55 nM
98%
Galeterone
++
Androgen Receptor, IC50: 384 nM
98%
Enzalutamide
+++
Androgen Receptor, IC50: 36 nM
98%
Megestrol
✔
98%
Bicalutamide
++
Androgen Receptor, IC50: 0.16 μM
99%
EPI-001
+
Androgen Receptor, IC50: ~6 μM
98%
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1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
N-Desmethyl-Apalutamide 实验方案
计算器
摩尔计算器
总药量计算器
工作液计算器
存储液制备
1mg
5mg
10mg
1 mM
5 mM
10 mM
2.16mL
0.43mL
0.22mL
10.79mL
2.16mL
1.08mL
21.58mL
4.32mL
2.16mL
N-Desmethyl-Apalutamide 技术信息
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