货号:A691315 同义名: (1R,2R)-2-PCCA hydrochloride
(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 agonist, with an EC50 of 3 nM.
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描述 | GPR88 is an orphan G-protein-coupled receptor that plays an essential role in regulating striatal functions. (1R,2R)-2-PCCA 2 is a potent GPR88 agonist that inhibits isoproterenol-induced cAMP formation with an EC50 value of 603nM (pEC50 = 6.22) in cell assay[1]. In CHO cells overexpressing the PPLS-HA-GPR88 construct, the EC50 value of (1R,2R)-2-PCCA 2 is 56nM[2]. |
计算器 | ||||
存储液制备 | 1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
1.89mL 0.38mL 0.19mL |
9.46mL 1.89mL 0.95mL |
18.92mL 3.78mL 1.89mL |
CAS号 | 1609563-71-4 |
分子式 | C30H39Cl2N3O |
分子量 | 528.556 |
别名 | (1R,2R)-2-PCCA hydrochloride |
运输 | 蓝冰 |
存储条件 |
粉末 Inert atmosphere,2-8°C 液体 -20°C:3-6个月-80°C:12个月 |
溶解度 |
DMSO: 50 mg/mL(94.6 mM),配合低频超声助溶,注意:DMSO长时间开封后,会吸水并导致溶解能力下降,请避免使用长期开封的DMSO |
动物实验配方 |