7ACC2 is a potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx for antitumor treatment targeting lactate transport in cancer cells.

VB124是一种 MCT4 抑制剂，具有高选择性，主要用于心脏肥大和代谢研究。

AZD0095是一种高选择性的口服活性 MCT4 抑制剂。它通过阻断乳酸转运，减少肿瘤细胞的乳酸排泄。与 Cediranib 联合使用时，AZD0095 显著抑制 NCI-H358 移植瘤的生长，展现出在抗肿瘤治疗中的潜力。

AZD3965 是一种选择性的乳酸转运体 1 (MCT1) 抑制剂，对 MCT1 具有高亲和力，IC50 值为 3 nM。AZD3965 具有抗肿瘤作用，可用于乳酸代谢相关癌症的研究。

BAY-8002 is a potent MCT Inhibitor with IC50 value of 8nM for inhibition of L-lactate uptake.

α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity.

7ACC1 selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment and inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters.

UK-5099 is a potent is MPC (mitochondrial pyruvate carrier) inhibitor with IC50 value of 50 nM.

Silychristin, a natural product isolated and purified from the herbs of Silybum marianum (L.) Gaertn., is a plant growth regulator, an anti-hepatotoxic agent, and an inhibitor of horseradish peroxidases and lipoxygenase.

SR13800 is a cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1).

AR-C155858 是一种选择性单羧酸转运蛋白 MCT1 和 MCT2 的抑制剂，Ki 分别为 2.3 nM 和 10 nM。