(2-Chloropyridin-4-yl)methanamine hydrochloride是一种选择性的 LOXL2 抑制剂，IC₅₀ 为 126 nM，适用于抗纤维化和癌症的研究。

PXS-5153A is a selective inhibitor of LOXL2 and LOXL3 with IC50 of <40 nM and 63 nM, respectively.

PAT-1251 is a potent, selective and oral Lysyl Oxidase-Like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively); PAT-1251 has entered clinical development with the potential to treat a number of fibrotic diseases.