ET-A

货号			产品名	纯度
A445755	现货	促	Zibotentan Zibotentan is an orally administered, potent and specific ETA-receptor (endothelin A receptor) antagonist (IC50 = 21 nM).	99%+
A404664	现货	促	Bosentan hydrate/波生坦水合物 Bosentan hydrate竞争性双重拮抗内皮素-1（ET）对ETA和ETB受体，在人体平滑肌细胞中Ki值分别为4.7 nM和95 nM。	98%
A539182	现货	促	Macitentan/马西替坦 Macitentan is an antagonist of endothelin receptor A (ETA) with IC50 of 0.5 nM. It is developed for treatment of pulmonary arterial hypertension (PAH).	98%
A121424	现货	促	Ambrisentan/安倍生坦 Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s = 0.251, 0.316, 0.398, 251, and 630 nM for rat preparations of heart, bladder, kidney, lung, and cerebral cortex, respectively).	98%
A370186			BQ-123 BQ-123 is a specific antagonist of endothelin A receptor (ETA) and the IC50 is 7.3 nM.	98%

货号

产品名

纯度

A445755

现货

促

Zibotentan is an orally administered, potent and specific ETA-receptor (endothelin A receptor) antagonist (IC50 = 21 nM).

99%+

A404664

现货

促

Bosentan hydrate/波生坦水合物

Bosentan hydrate竞争性双重拮抗内皮素-1（ET）对ETA和ETB受体，在人体平滑肌细胞中Ki值分别为4.7 nM和95 nM。

98%

A539182

现货

促

Macitentan/马西替坦

Macitentan is an antagonist of endothelin receptor A (ETA) with IC50 of 0.5 nM. It is developed for treatment of pulmonary arterial hypertension (PAH).

98%

A121424

现货

促

Ambrisentan/安倍生坦

Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s = 0.251, 0.316, 0.398, 251, and 630 nM for rat preparations of heart, bladder, kidney, lung, and cerebral cortex, respectively).

98%

A370186

BQ-123

BQ-123 is a specific antagonist of endothelin A receptor (ETA) and the IC50 is 7.3 nM.

98%