Mtb ATP synthase-IN-1是一种高效的抗结核分枝杆菌 ATP 合成酶抑制剂，MIC 值为 0.452-0.499 μg/mL，显示出良好的代谢稳定性和低细胞毒性。该化合物具有良好的口服生物利用度，适用于抗结核的研究。

Bedaquiline, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections.

Oligomycin A, a mitochondrial ATP synthase inhibitor, is isolated from Streptomyces species, exhibits anti-tumor and antibiotic activity.

BTB06584 is an IF1-dependent selective inhibitor of the mitochondrial F1Fo-ATPase.

Bedaquiline fumarate, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections.

D-α-Hydroxyglutaric acid是神经代谢疾病 D-2-羟基戊二酸尿症的主要代谢产物，能够抑制多种 α-酮戊二酸依赖性双加氧酶，Ki 为 10.87 mM，同时通过增加 ROS 生成抑制 ATP 合酶并抑制 mTOR 信号通路，适用于代谢及神经疾病研究。

PD173952 是一种酪氨酸激酶抑制剂，其对 Lyn、Abl 和 Csk 的 IC50 值分别为 0.3 nM、1.7 nM 和 6.6 nM。它也是 Myt1 的抑制剂，Ki 为 8.1 nM，并可诱导细胞凋亡。

ZW290是一种能够激活棕色脂肪组织 (BAT) 生热功能的化合物，能显著增加 BAT 中解偶联蛋白 1 (UCP1) 的表达，并抑制 ATP 合成，具有调节能量代谢的潜力。

Bz 423 is an ATP synthase inhibitor woth IC50 ~5 μM.

Oligomycin Complex is a mixture of oligomycins A, B, and C. Oligomycin A is a selective inhibitor of mitochondrial F1FO-ATP synthase that induces apoptosis in a variety of cell types. Oligomycin B is a nonselective inhibitor of ATP synthases. Oligomycin B can reduce the rate of ATP depletion in myocardial ischemia and decrease calcium-induced calcium release oscillation frequency of rat sensory neurons.