Actinonin is a bioactive peptide and antibiotic that is a potent inhibitor of CD13 and aminopeptidase (leucine aminopeptidase).

Aminopeptidase-IN-1是一种胰岛素调节氨肽酶 (IRAP) 的有效抑制剂，Ki 为 7.7 μM。该化合物可用于认知和记忆障碍的研究，具有开发治疗阿尔茨海默病和其他神经退行性疾病的潜力。

Tosedostat is a aminopeptidase inhibitor with IC50 of 220, > 1000 nM for aminopeptidase N and aminopeptidase B respectively.

SC-57461A is a selective inhibitor of LTA4H (leukotriene A4 hydrolase).

LTA4H-IN-1是一种高效的白三烯 A4 水解酶 LTA4H 抑制剂，IC50 值为 2 nM，可用于炎症和自身免疫性疾病的研究。

Bestatin is a competitive and specific inhibitor of leucine aminopeptidase, aminopeptidase B, and triamino peptidase.

Bestatin HCl is a competitive and specific inhibitor of leucine aminopeptidase, aminopeptidase B, and triamino peptidase.

L-Leucine-p-nitroanilide is a leucine aminopeptidase substrate.

TNP-470, a synthetic analogue of fumagillin and an antiangiogenic compound, is inhibitor of methionine aminopeptidase-2 (MetAP-2) and can inhibit angiogenesis.