GW406108X(Z/E)是一种具有生物活性的化合物，主要作为Kif15（Kinesin-12）的特异性抑制剂。它还显示出对ULK1（Unc-51 like kinase 1）的ATP竞争性抑制作用，

Litronesib is a selective, allosteric inhibitor of Eg5, which may result in mitotic disruption, apoptosis and consequently cell death in tumor cells that are actively dividing.

GSK-923295 是一种特异性的着丝粒相关蛋白 E (CENP-E) 驱动蛋白 ATP 酶活性的变构抑制剂，对人和犬的 Ki 值分别为 3.2±0.2 nM 和 1.6±0.1 nM。

SB-743921 is a potent KIF11 inhibitor with Ki value of 0.1 nM.

Filanesib hydrochloride是一种 Kinesin spindle protein (KSP) 抑制剂，能够干扰细胞分裂。它在癌症治疗中展现出显著的抗增生活性。

Monastrol is a specific and allosteric inhibitor of mitotic molecular motor kinesin Eg5 with IC50 value of 14 μM.

BRD9876 is a selective inhibitor of MM1S growth. It is selective for microtubule bound Eg5 and causes a rapid arrest in G2/M phase.

Ispinesib is a quinazolinone-derived, specific and reversible kinesin spindle protein inhibitor with Ki_app value of 1.7 nM.

AZ3146 is a selective and potent Mps1 inhibitor with IC50 value of 35 nM.

MPI-0479605 is a potent and selective ATP competitive Mps1 with IC50 value of 1.8 nM.

H-Cys(Trt)-OH is a potent and selective inhibitor of mitotic kinesin Eg5 with IC50 value of 140 nM.