PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.

T863 is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA binding site of DGAT1, and inhibits triacylglycerol synthesis in cells.

LCQ-908 is a potent and oral active diacylglycerol acyltransferase 1 (DGAT1) inhibitor, used as anti-obesity and anti-diabetic agents.

PF-07202954是一种弱碱性 DGAT2 抑制剂，对人 DGAT2 的 IC₅₀ 为 10 nM。该化合物在降低脂肪积累、调节脂质代谢及心血管疾病研究中展示了显著的作用，适用于脂肪肝和相关疾病的研究。

Etomoxir is a cell-permeable, irreversible, and stereospecific inhibitor of carnitine palmitoyltransferase (CPT)-1 and DGAT activity in the mitochondria of rat heart H9c2 myoblastic cells at a concentration of 1-80 μM and 40 μM, respectively.

A 922500（DGAT-1抑制剂4a）是一种强效、选择性和口服生物利用度的甘油二酰基转移酶1（DGAT-1）抑制剂，其对人类和小鼠DGAT-1的IC50值分别为9 nM和22 nM。

Ervogastat is a diacylglycerol acyltransferase type 2 (DGAT-2) inhibitor.

DGAT1-IN-1 is a potent DGAT1 inhibitor with IC50 of < 10 nM (cell lysate from Hep3B cells overexpressing human DGAT1).

Teglicar (ST-1326) is a potent, selective and reversible inhibitor of liver carnitine palmitoyl-transferase 1 (L-CPT1) with IC50 of 0.68 uM, Ki of 0.36 uM.

AZD7687 is a potent and selective DGAT1 inhibitor with an IC50 of 80 nM for hDGAT1.

Aphadilactone C is a naturla product isolated and purified from Aphanamixis grandifolia with DGAT inhibitory and antimalarial activities.

DGAT-1 inhibitor 2 is an effective inhibitor of DGAT-1 and an antiobesity agent.