Vazegepant是一种高效、选择性且结构独特的小分子 CGRP 受体拮抗剂。

Rimegepant是一种高效口服降钙素基因相关肽（CGRP）受体拮抗剂，Ki 值为 0.027 nM。

Galcanezumab是一种人源化IgG4单克隆抗体，通过与CGRP结合来阻止其与受体结合。Galcanezumab具有用于偏头痛预防的潜力。

α-CGRP(8-37), huma is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor.

Rat CGRP-(8-37) is a highly selective antagonist of CGRP receptor.

Ubrogepant is an oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine.

Calcitonin salmon is a calcium regulating hormone secreted from mammalian thyroid parafollicular cells and in non-mammalian species from the ultimobranchial gland.

Fremanezumab是一种人源化IgG2单克隆抗体，通过与CGRP结合来阻止其与受体结合。Fremanezumab具有用于偏头痛预防的潜力。

MK-3207是一种强效且口服有效的 CGRP 受体拮抗剂，IC50 为 0.12 nM，Ki 值为 0.024 nM，对人类 AM1、AM2、CTR 和 AMY3 具有高度选择性。

SUN-B 8155 is a non-peptide calcitonin agonist.