Scutellarin is cytotoxic to cancer cells and could induce DNA damage, metabolic suppression and mitochondrial reactive oxygen species. It has has antioxidant, anti-inflammatory, and antiproliferative biological activities that can be can be found in scutellaria lateriflora.

Scutellarein tetramethyl ether是从 Eupatorium odoratum 提取的生物活性成分，通过 NF-κB 通路发挥抗炎作用。此外，它通过外排泵抑制作用调节细菌耐药性，并能增强凝血功能。

Oroxin B, a natural product isolated and purified from the roots of Scutellaria baicalensis., can selectively induce tumor-suppressive ER stress and concurrently inhibit tumor-adaptive ER stress in B-lymphoma cells for effective anti-lymphoma therapy.

Wogonin 是一种天然黄酮类化合物，能够抑制 CDK8 和 Wnt 的活性。Wogonin 具有抗炎和抗肿瘤的功效，主要用于抗炎症和抗癌研究。

Oroxin A is the major component of an ethanol-water Oroxylum indicum (L.) Kurz (Bignoniaceae) seed extract (OISE), activates peroxisome proliferator-activated receptor γ (PPARγ) by docking into the PPARγ protein ligand-binding domain. Oroxin A exhibits an inhibitory activity against α-glucosidase and an antioxidant capacity. Oroxin A exerts anti-breast cancer effects by inducing ER stress-mediated senescence.

Plantagoside是一种从 Plantago asiatica 中提取的 α-mannosidase 抑制剂，具有选择性和非竞争性抑制作用。它在糖尿病和与糖代谢相关的疾病研究中展现了应用前景。

Wogonoside is a natural product isolated and purified from the herbs of Scutellaria baicalensis Georgi.

5,6,7-Trimethoxyflavone是一种 p38 MAPK 抑制剂，具有显著的抗炎作用。它通过干扰 p38 MAPK 信号通路，对多种炎症相关疾病和肿瘤模型中展现出治疗潜力。

Oroxylin A 7-O-beta-D-glucuronide, a natural product isolated and purified from the roots of Scutellaria regeliana Nakai., can bind to the "stem" region of α-hemolysin (α-HL), when inhibiting the hemolytic activity of α-HL, and inhibit 34% of total prolyl oligopeptidase (POP) activity, respectively at a concentration of 100 mM.

Ombuoside has antifungal activity. Ombuoside shows significant antioxidant activity in the DPPH, and TEAC, reducing power assays.

5,7,8-Trimethoxyflavone是一种来自穿心莲的黄酮类化合物，具有抗炎特性，能够抑制一氧化氮 (NO) 生成，IC₅₀ 为 39.1 μM。

Scutebarbatine A, a natural product isolated and purified from the herbs of Scutellaria barbata D. Don, shows significant antitumor effects on A549 cells in vivo and in vitro via mitochondria-mediated apoptosis by up-regulating expressions of caspase-3 and 9, and down-regulating Bcl-2, and a significant ability to protect cells against H2O2 with ED50 values of 5.0 and 16.8 uM, respectively.

Skullcapflavone I, a natural product isolated and purified from the roots of Scutellaria baicalensis Georgi, selectively induces apoptosis in T-HSC/Cl-6 cells via caspase-3 and caspase-9 activation.

4'-Hydroxywogonin, a natural product isolated and purified from the roots of Scutellaria baicalensis Georgi, has positive effect on inhabiting those human tumor lines in vitro, with IC50 value is 8.3-38.4 ug/mL .

Apigenin 5-O-beta-D-glucopyranoside is a natural product isolated and purified from the herbs of Scutellaria barbata with inhibitory activity against the enzyme yeast a-glucosidase, the IC50 values 287.12 μM.