LM11A-31 2HCl是一种非肽 p75NTR（神经营养蛋白受体 p75）调节剂，作为口服有效的 proNGF 拮抗剂，具有良好的血脑屏障通透性，能阻断 p75 介导的细胞死亡。

SBI-553是一种有效且可穿透大脑的 NTR1 的变构调节剂，EC50 为 0.34 μM。

ML314是NTR1的强效分子激动剂（EC50 = 1.9 μM），对NTR2和GPR35具有良好的选择性，但未能刺激Ca2+动员。

PD 90780 is a non-peptide inhibitor of nerve growth factor (NGF) binding to p75NTR receptor. It inhibits NGF-p75 NTR interaction with IC50s values of 23.1 µM and 1.8 µM in PC12 cells and PC12 nnr5 cells, respectively.

Neurotensin, a potent hypothalamic peptide neurotransmitter, is an endogenous anti-psychotic compound which has a high affinity for neurotensin receptors.

JMV 449 is a potent, metabolically stable neurotensin receptor agonist peptide.

Kinetensin is endogenous neurotensin-like peptide originally isolated from pepsin-treated human plasma. It can induce histamine release from rat peritoneal mast cells in vitro.

Neurotensin Fragment 8-13 is the smallest active fragment of neurotensin which is a potent cellular mitogen for various colorectal and pancreatic cancers which possess high-affinity neurotensin receptors (NTR).

Xenopsin is the neurotensin-like octapeptide from Xenopus skin at the carboxyl terminus of its precursor.