Seneciphylline是从 Senecio scandens（藤本金露梅）草本植物中分离和纯化的天然产物，能够显著增加环氧化酶和谷胱甘肽-S-转移酶的活性，但导致细胞色素 P-450 及相关单加氧酶活性减少。

GSTO1-IN-1是一种强效的谷胱甘肽S-转移酶ω1（GSTO1）抑制剂，IC50值为31 nM。

Ezatiostat是谷胱甘肽的类似物，能够抑制谷胱甘肽S-转移酶P1-1（GSTP1-1）。

trans-Methylisoeugenol是一种天然食用香料，具有抗焦虑和抗抑郁作用，可抑制谷胱甘肽S-转移酶的活性。

Coniferyl ferulate is a natural product.

GSTO-IN-2 is a glutathione S-transferase inhibitor with IC50s of 3.6, 16.3, and 1.4 μM for GSTA2, GSTM1, and GSTP1-1.

3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid is a natural product isolated and purified from the barks of Caesalpinia bonduc with glutathione S-transferase (GST) inhibitory and antifungal activities.

Ezatiostat HCl is a glutathione analog inhibitor of glutathione S-transferase P1-1 (GSTP1-1).