Brevifolincarboxylic acid 是从蓼属植物提取的，对芳烃受体 (AhR) 有抑制作用，也是 α-葡萄糖苷酶的抑制剂，IC50 值为 323.46 μM。

GCase modulator-1是一种 Quinolazoline 衍生物，作为葡萄糖苷酶 (GCase) 的调节剂，具有 AC50 值为 2.23 μM 的活性。该化合物适用于溶酶体贮积病和与 GCase 功能相关的疾病的研究。

NCGC 607是葡萄糖脑苷酶 (Gcase) 的非抑制性分子伴侣，主要用于研究特定的酶抑制机制和与代谢疾病相关的信号通路。

Butyl isobutyl phthalate is isolated from the rhizoid of Laminaria japonica. Butyl isobutyl phthalate is a non-competitive α-glucosidase inhibitor with an IC50 value of 38 μM. Butyl isobutyl phthalate shows a hypoglycemic effect and has the potential for diabetes treatment.

3,4-Dicaffeoylquinic Acid is a polyphenol with diverse biological activities, it inhibits acetylcholinesterase (ACE) and α-glucosidase in a concentration-dependent manner, shows cytotoxic to NCI-H23 lung adenocarcinoma cells, as well as increases tumor necrosis factor-related apoptosis inducing ligand (TRAIL) mRNA, reduces influenza H1N1 hemagglutinin (HA) mRNA and increases survival in a mouse model of influenza A infection.

7,4'-Di-O-methylapigenin, a flavonoid purified from aquilaria sinensis, can inhibit α-glucosidase, α-amylase enzymes and enhance 2-NBDG uptake in L6 cells. It has hypolipidemic effect.

Miglitol is a desoxynojirimycin-derived inhibitor of alpha-glucosidase with antihyperglycemic activity.

Voglibose, an N-substituted derivative of valiolamine, can inhibit α-glucosidase and be used to treat hyperglycemia and its concomitant diseases.

2'-Methoxykurarinone, a natural product isolated and purified from the roots of Sophora flavescens Ait.

ML198是一种用于戈谢病研究的葡萄糖脑苷脂酶 (GCase) 调节剂。它也可用于点击化学试剂，具有非抑制性伴侣的特性。

Demethylisoencecalin 属于黄酮类化合物，通常从植物中提取，具有抗炎、抗氧化和抗肿瘤等生物活性。Demethylisoencecalin 是一种有效的 α-葡萄糖苷酶抑制剂，IC50 值为 0.169 mg/mL。

α-Glucosidase-IN-22是一种苯并咪唑类 α-葡萄糖苷酶 (α-glucosidase) 抑制剂，IC₅₀ 为 0.64 μM，显示出强效的抗糖尿病活性，具有在 2 型糖尿病研究中的应用潜力。

Licochalcone C 以 <100 nM 的 IC50 值抑制 α-葡萄糖苷酶，以 92.43 μM 的 IC50 值抑制蛋白酪氨酸磷酸酶 1B。

Kaempferol 7-O-rhamnoside is a natural product isolated and purified from the herbs of Maytenus hookeri.

Castanospermine inhibits all forms of α- and β-glucosidases, especially glucosidase l (required for glucoprotein processing by transfer of mannose and glucose from asparagine-linked lipids).

Methyl caffeate is an α-glucosidase inhibitor found in species of Solanum and Magnolia. It exhibits several biological activities, including suppressing growth of Pseudomonas, Klebsiella, and Mycobacterium, inhibiting replication of HIV, and decreasing blood glucose levels in models of diabetes.

ML266 is a glucocerebrosidase activator and a non-inhibitory chaperone of glucocerebrosidase.

Deoxynojirimycin HCl, a natural product isolated and purified from the root barks of Morus alba L., shows inhibitory activity against α-glucosidases, inhibitors of α-glucosidase are promising candidates for the development of antitype II diabetics and anti-AIDS drugs.

N-Nonyldeoxynojirimycin is a glucosidase inhibitor with IC50s of 0.42 and 8.4 μM for acid α-glucosidase and α-1,6-glucosidase respectively.

N-Methylmoranoline is an inhibitor of α-glucosidase inhibitor.