WAY-213613 hydrochloride是一种有效的、选择性人EAAT2抑制剂，IC₅₀值为85 nM，常用于中枢神经系统相关疾病的研究，特别是在神经退行性疾病中的应用。

DL-TBOA is a competitive and non-transportable blocker of excitatory amino acid transporters with IC50 values of 70, 6, 6, 4.4 and 3.2 μM for EAAT1, EAAT2, EAAT3, EAAT4 and EAAT5 respectively.

WAY-213613 is a potent, selective GLT-1/EAAT2 (functional glutamate transporter/excitatory amino acid transporter) nonsubstrate inhibitor with IC50s of 85 nM, 5 μM and 3.8 μM for EAAT2, EAAT1 and EAAT3. WAY-213613 is a highly EAAT2-preferring transporter ligand and inhibits glutamate uptake in rat cortical synaptosomes[1][2].