BRD2/PROTAC

货号	产品名	纯度
A482817	PROTAC BET Degrader 9 PROTAC BET degrader-9 is PROTAC targeting on BET proteins, consist of a BET inhibitor HJB97 as the warhead ligand and Pomalidomide as CRBN ligand.	98%
A1554996	MS83	98+%
A1553215	PROTAC BRD2/BRD4 degrader-1	98%
A376159	MZP-54 MZP-54 is a PROTAC targeting on BET, consist of a warhead I-BET726 (BET bromodomain inhibitor) linked to a VHL ligand VH032.	98%
A176034	MZP-55 MZP-55 is a VHL-based PROTAC targeting on BET with pDC₅₀/D_max (%) values of 8.1/95, 7.5/93, 7.7/92, −/26 for Brd4 short, Brd4 long, Brd3 and Brd2 in HeLa cells, consist of I-BET726 as a warhead ligand linked to VHL ligand VH032.	98%

货号

产品名

纯度

A482817

PROTAC BET degrader-9 is PROTAC targeting on BET proteins, consist of a BET inhibitor HJB97 as the warhead ligand and Pomalidomide as CRBN ligand.

98%

A1554996

MS83

98+%

A1553215

PROTAC BRD2/BRD4 degrader-1

98%

A376159

MZP-54

MZP-54 is a PROTAC targeting on BET, consist of a warhead I-BET726 (BET bromodomain inhibitor) linked to a VHL ligand VH032.

98%

A176034

MZP-55

MZP-55 is a VHL-based PROTAC targeting on BET with pDC₅₀/D_max (%) values of 8.1/95, 7.5/93, 7.7/92, −/26 for Brd4 short, Brd4 long, Brd3 and Brd2 in HeLa cells, consist of I-BET726 as a warhead ligand linked to VHL ligand VH032.

98%