Apelin-13 TFA是 G 蛋白偶联受体angiotensin II protein J (APJ) 的内源性配体，激活G蛋白偶联受体的 EC50 值为 0.37 nM。Apelin-13 TFA 具有扩张血管和降压作用。Apelin-13 TFA 也可用于 2 型糖尿病及代谢综合征的研究。

ML221是一种强效 apelin 受体（APJ）拮抗剂，在 cAMP 和 β-arrestin 实验中的 IC50 分别为 0.70 μM 和 1.75 μM，选择性高于 AT1 受体。

Saikogenin A, extracted from a Chinese herbal plant called Tsai-Fu, is a dipeptidyl peptidase-IV (DPP-IV) inhibitor.

CY3-SE is a reactive dye for the labeling of amino-groups in biomolecules.

Demethylzeylasteral, a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f., has strong immunosuppressive activity, that can be used in the fields of organ transplantation and autoimmune disorders. It increases both activation and inactivation time constants of Ca(2+) currents, and inhibits significantly the sperm acrosome reaction initiated by progesterone.

[Pyr1]-Apelin-13是一种高效的肽 Apelin 激动剂，EC50 为 0.37 nM。

NRX-103094, a molecular glue, is a potent enhancer of the interaction between β-catenin, and its cognate E3 ligase, SCFβ-TrCP. NRX-103094 enhances the binding of pSer33/Ser37 β-catenin peptide for β-TrCP with an EC50 of 62 nM and a Kd of 0.6 nM.