Apelin-13 TFA是 G 蛋白偶联受体angiotensin II protein J (APJ) 的内源性配体，激活G蛋白偶联受体的 EC50 值为 0.37 nM。Apelin-13 TFA 具有扩张血管和降压作用。Apelin-13 TFA 也可用于 2 型糖尿病及代谢综合征的研究。

ML221是一种强效 apelin 受体（APJ）拮抗剂，在 cAMP 和 β-arrestin 实验中的 IC50 分别为 0.70 μM 和 1.75 μM，选择性高于 AT1 受体。

Azelaprag 是一种 apelin 受体激动剂的候选活性分子，可用于治疗神经系统疾病和心血管疾病。

Schisandrin C is a phytochemical lignan isolated from Schizandra chinensis Baill and shows anticancer-effects in human leukemia U937 cells.

ML339 是一种选择性的 CXCR6 拮抗剂，IC50 为 140 nM。它对 CXCL16 诱导的人 CXCR6 受体的 β-阻滞蛋白募集和 cAMP 信号通路有拮抗作用，IC50 分别为 0.3 μM 和 1.4 μM。ML339 对小鼠 CXCR6 受体上拮抗 β-阻滞蛋白募集的活性较弱，IC50 为 18 μM。ML339 对 CXCR5、CXCR4、CXCR6 和 Apelin 受体 (APJ) 无抑制作用，IC50 >79 μM。

Saikogenin A, extracted from a Chinese herbal plant called Tsai-Fu, is a dipeptidyl peptidase-IV (DPP-IV) inhibitor.

CY3-SE is a reactive dye for the labeling of amino-groups in biomolecules.

Demethylzeylasteral, a natural product isolated and purified from the herb of Tripterygium wilfordii Hook.f., has strong immunosuppressive activity, that can be used in the fields of organ transplantation and autoimmune disorders. It increases both activation and inactivation time constants of Ca(2+) currents, and inhibits significantly the sperm acrosome reaction initiated by progesterone.