生物活性 | |||
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描述 | Similarly, CB2R/FAAH modulator-3 is characterized as a dual targeting modulator acting as a CB2R agonist and FAAH inhibitor. It exhibits Ki values of 20.1 nM and 67.6 nM for CB2R and CB1R, respectively, and an IC50 value of 3.4 μM for FAAH. CB2R/FAAH modulator-3 also shows potential for use in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection [1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
2.93mL 0.59mL 0.29mL |
14.64mL 2.93mL 1.46mL |
29.28mL 5.86mL 2.93mL |
参考文献 |
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