生物活性 | |||
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描述 | MS48107 is a potent and selective positive allosteric modulator of G protein-coupled receptor 68 (GPR68). It shows selectivity for GPR68 over closely related proton GPCRs, neurotransmitter transporters, and hERG ion channels. MS48107 can effectively cross the blood-brain barrier (BBB) in mice[1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
2.40mL 0.48mL 0.24mL |
11.98mL 2.40mL 1.20mL |
23.96mL 4.79mL 2.40mL |
参考文献 |
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