产品说明书

(E/Z)-Ensifentrine

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Chemical Structure| 298680-25-8 同义名 : (E/Z)-RPL-554
CAS号 : 298680-25-8
货号 : A982733
分子式 : C26H31N5O4
纯度 : 99%+
分子量 : 477.555
MDL号 : N/A
存储条件：

粉末 Sealed in dry,Store in freezer, under -20°C

液体 -20°C:3-6个月-80°C:12个月
溶解度 : -
动物实验配方：
生物活性
描述 (E/Z)-Ensifentrine is a dual inhibitor of PDE3/4. (E/Z)-Ensifentrine reduces inflammatory cells entering the respiratory tract. (E/Z)-Ensifentrine has bronchodilatory and anti-inflammatory activity in both in vitro and in vivo models[1].
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.09mL

0.42mL

0.21mL

10.47mL

2.09mL

1.05mL

20.94mL

4.19mL

2.09mL
参考文献

[1]Page CP, et al. Phosphodiesterase inhibitors for the treatment of asthma and chronic obstructive pulmonary disease. Int Arch Allergy Immunol. 2014;165(3):152-64.