Selurampanel

产品说明书

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Chemical Structure| 912574-69-7 同义名 : BGG 492
CAS号 : 912574-69-7
货号 : A813453
分子式 : C16H19N5O4S
纯度 : 99+%
分子量 : 377.418
MDL号 : -
存储条件：

Pure form

In solvent -20°C:3-6个月-80°C:12个月
溶解度 : -
动物实验配方：
生物活性
描述 Selurampanel is a competitive AMPA/kainate receptor antagonist drug for epilepsy.
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.65mL

0.53mL

0.26mL

13.25mL

2.65mL

1.32mL

26.50mL

5.30mL

2.65mL
参考文献

[1]Orain D, Tasdelen E, et al. Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist. ChemMedChem. 2017 Feb 3;12(3):197-201.

[2]Faught E. BGG492 (selurampanel), an AMPA/kainate receptor antagonist drug for epilepsy. Expert Opin Investig Drugs. 2014 Jan;23(1):107-13.