生物活性 | |||
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描述 | (E/Z)-GSK-3β inhibitor 1 is a racemic mixture composed of the (E)-GSK-3β inhibitor 1 and (Z)-GSK-3β inhibitor 1 isomers. It functions as an inhibitor of glycogen synthase kinase 3β (GSK-3β) and exhibits significant antidiabetic efficacy, with an IC50 value of 4.9 nM[1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
4.50mL 0.90mL 0.45mL |
22.50mL 4.50mL 2.25mL |
45.00mL 9.00mL 4.50mL |
参考文献 |
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