生物活性 | |||
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描述 | S-methyl-KE-298 is the methyl conjugate of deacetyl-KE-298 in plasma[1]. In vitro protein binding of KE-298 and its plasma metabolites, deacetyl-KE-298 (M-1) and S-methyl-KE-298 (M-2), is greater than 97% in rats, over 89% in dogs, and more than 99% in human plasma[2]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
3.96mL 0.79mL 0.40mL |
19.82mL 3.96mL 1.98mL |
39.63mL 7.93mL 3.96mL |
参考文献 |
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