GSK-2881078

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Chemical Structure| 1539314-06-1 同义名 : -
CAS号 : 1539314-06-1
货号 : A275241
分子式 : C14H13F3N2O2S
纯度 : 98+%
分子量 : 330.325
MDL号 : MFCD30343844
存储条件：

Pure form Sealed in dry,Store in freezer, under -20°C

In solvent -20°C:3-6个月-80°C:12个月
溶解度 :

DMSO: 35 mg/mL(105.96 mM)，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO
动物实验配方：
生物活性
描述 GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia.
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

3.03mL

0.61mL

0.30mL

15.14mL

3.03mL

1.51mL

30.27mL

6.05mL

3.03mL
参考文献

[1]Clark RV, Walker AC, et al. Safety, pharmacokinetics and pharmacological effects of the selective androgen receptor modulator, GSK2881078, in healthy men and postmenopausal women. Br J Clin Pharmacol. 2017 Oct;83(10):2179-2194.